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1-[4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(1H-1,2,4-triazol-3-ylsulfanyl)ethan-1-one
3-(azocan-1-yl)-N-[(4-fluorophenyl)methyl]-N-methylpropanamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxamide
2-[3-cyclopentyl-5-(2,3-dihydro-1-benzofuran-2-yl)-1H-1,2,4-triazol-1-yl]acetic acid
(3R,5S)-N3-(4-fluorophenyl)-N5-(3-methoxypropyl)-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
2-(2-ethyl-1H-imidazol-1-yl)-1-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
2-[(1-methylpiperidin-4-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
6-{1-[(3-chloro-4-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]acetamide
2,6-dimethyl-3-[4-(pyridin-4-yl)piperazine-1-carbonyl]quinoline
1-(2,3-dimethylquinoxalin-6-yl)-3-[3-(1H-1,2,3-triazol-1-yl)propyl]urea
1-(3-methyl-1H-pyrazole-4-carbonyl)-4-[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]piperidine
6-{[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]methyl}-2-methylpyrimidin-4-ol
8-benzoyl-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(1,4-dithiepan-6-yl)piperazin-2-yl}ethan-1-ol
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(6-methylpyridin-2-yl)piperazine
N-cyclopropyl-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}oxolane-2-carboxamide
3-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)-1-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]phenyl}urea
2-(4-methanesulfonylphenyl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
1-{3-[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]propyl}pyrrolidin-2-one
(1R,7S)-3-(2-methoxyethyl)-6-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
6-(3-fluorophenyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-({3-[4-(difluoromethoxy)phenyl]phenyl}methyl)morpholine
5-(ethylsulfanyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]thiophene-2-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-3-(1H-pyrazol-1-yl)benzamide
4-{1-[1-(pyrazin-2-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
ethyl 1-{3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanoyl}piperidine-2-carboxylate
(5S,9aS,9bS)-5-(4-hydroxy-3,5-dimethylphenyl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}-N-methylpyrrolidine-3-carboxamide
2-(2-ethoxyphenyl)-2-[4-(furan-2-carbonyl)piperazin-1-yl]acetic acid
2-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
(3aR,6aR)-2-cyclopentyl-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aS,8aR)-1-(2-aminoethyl)-6-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-decahydro-1,6-naphthyridin-2-one
2-methyl-4-{3-[(2S)-4-methyl-2-phenylpiperazine-1-carbonyl]phenyl}butan-2-ol
5-(2-{[(4-fluorophenyl)methyl](methyl)amino}acetyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
5-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-2,4-dimethyl-1,3-oxazole
8-[(2-fluoro-4-methylphenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
4-({4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)-1-methylpyrrolidin-2-one
1-benzyl-N3-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(2R)-N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]oxolane-2-carboxamide
(1R,5S,8R)-3-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-3-azabicyclo[3.2.1]octan-8-ol
N-[1-(4-methoxyphenyl)ethyl]-N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetamide
1-{2-oxo-2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
3-[(cyclohexylamino)methyl]-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
N-ethyl-N-[1-(4-methoxyphenyl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(2-ethoxypyridin-3-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-[(3-methylphenyl)methyl]-4-[3-(methylsulfanyl)butyl]piperazine
2-(2-fluoro-5-methoxyphenyl)-2-[(2-methoxyethyl)(methyl)amino]acetic acid
2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoline