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1-(4-benzylpiperidin-1-yl)-3-[1-(2-hydroxy-6-methylpyridine-3-carbonyl)piperidin-4-yl]propan-1-one
1-cycloheptyl-N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-6-oxopiperidine-3-carboxamide
5-methyl-1-(4-methylphenyl)-4-(quinoline-4-carbonyl)piperazin-2-one
3-(4-chloro-2-methylbenzoyl)-1-(4-methoxybenzoyl)piperidine
methyl 1-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxylate
8-[(2,3-dimethoxyphenyl)methyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-cyclopentyl-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-{4-[(2-aminopyridin-3-yl)methyl]morpholin-3-yl}-N-(pyridin-2-ylmethyl)acetamide
1-(3,4-dichlorophenyl)-4-(oxane-4-carbonyl)piperazine
2-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-pyrrol-1-yl)-4-methylpyridine
N-methyl-1-phenyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazole-5-carboxamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]pent-4-enamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
3-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-N-methylbutanamide
4-ethyl-3-[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2-methylphenyl)-2-[(1-phenoxypropan-2-yl)amino]acetamide
2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]acetamide
N-[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
4-{2-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-2-oxoethyl}-7-methyl-2H-chromen-2-one
4-(4-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
(1S,5R)-3-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-(1-{1-[(2-chloro-3,6-difluorophenyl)methyl]piperidin-4-yl}ethyl)-4-methylpiperazine
1-{3-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]phenyl}ethan-1-one
6-oxo-1-(3-phenylpropyl)-N-{2-[4-(trifluoromethyl)phenyl]ethyl}piperidine-3-carboxamide
3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-one
methyl 5-{[1-(4-fluorophenyl)propan-2-yl]amino}-1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[(4-benzyl-1H-1,2,3-triazol-1-yl)methyl]-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine
2-(dimethylamino)-2-(4-methylphenyl)-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]acetamide
N-{2-[(5-methyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}phenyl)formamido]ethyl}acetamide
ethyl 1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylate
8-[(1R,2R,3S,4S)-3-aminobicyclo[2.2.1]heptane-2-carbonyl]-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-ethyl-4-(1H-pyrazol-3-yl)phenyl]acetamide
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]quinoxaline-5-carboxamide
6-[5-(methoxymethyl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]-2-methyl-1,3-benzothiazole
3-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-N,N-dimethylaniline
N-(3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}phenyl)pentanamide
4-(5-methyl-1,3,4-oxadiazol-2-yl)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
4-{[3-(2-hydroxyethoxy)phenyl]methyl}-5-methyl-1-(4-methylphenyl)piperazin-2-one
2-(4-fluorophenoxymethyl)-4-hydroxy-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]pyrimidine-5-carboxamide
2-[(4aR,7aS)-6,6-dioxo-4-[2-(propan-2-yloxy)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
4-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)butanamide
N-butyl-N-methyl-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
3-(dimethylsulfamoyl)-5-{[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]amino}-N-[(1R)-1-(4-methoxyphenyl)ethyl]benzamide
(1R,5S,6S)-6-[3-(2-phenylethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-3-azabicyclo[3.1.0]hexane
2-amino-6-(2,2-dimethylcyclopropyl)-4-(1H-imidazol-4-yl)-5-methylpyridine-3-carbonitrile
3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-5-(5-methylfuran-2-yl)-1,2,4-triazine
1-{4-methyl-2-[methyl(quinoxalin-2-ylmethyl)amino]pyrimidin-5-yl}ethan-1-one