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1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
methyl 3-(2-ethoxypyridin-3-yl)benzoate
N4,N4,N6-trimethyl-N6-[(5-methyl-1H-pyrazol-3-yl)methyl]pyrimidine-4,6-diamine
6-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
(1R,7S)-3-tert-butyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-{3-[4-({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}amino)piperidin-1-yl]phenyl}pyrrolidin-2-one
1-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
2-[4-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)piperazin-1-yl]pyrazine
3-(4-chloro-3-fluorophenyl)-1,2,4,5,10,11-hexaazatricyclo[7.3.0.02,6]dodeca-3,5,7,9,11-pentaene
(1S,5R)-3-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-benzyl-2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)morpholine
N-{1-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetyl]pyrrolidin-3-yl}acetamide
(3S,4R)-3-methoxy-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-4-amine
6-(4-fluorophenyl)-N-methyl-N-(2-methylprop-2-en-1-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-acetyl-N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]thiophene-3-carboxamide
(3aS,6aR)-5-(4,6-dimethoxypyrimidin-2-yl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(4-ethylpiperazin-1-yl)-3-[2-methoxy-4-({[(3-methoxyphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
2,5-dimethyl-3-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
1-phenyl-3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}pyrrolidin-2-one
4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidine
2-(3-methyl-1,2-oxazol-5-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)acetamide
5-(methoxymethyl)-N-[(7-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]furan-2-carboxamide
methyl (2S,4S)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-[3-(4-methylphenyl)propanamido]pyrrolidine-2-carboxylate
(3aS,6aS)-2-(2-methoxyethyl)-5-[2-(6-methylpyridin-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(furan-3-ylmethyl)pyrrolidin-3-yl]-2-methyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-({[(5-methylthiophen-2-yl)methyl]amino}methyl)piperidin-2-one
(1-{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}-2,5-dihydro-1H-pyrrol-2-yl)methanol
2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-6-(4H-1,2,4-triazol-4-yl)pyridine
2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-ethylacetamide
(4aR,7aS)-1-butanoyl-4-(2-chlorobenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N,6-dimethylpyrimidin-2-amine
1-[(1-ethyl-1H-pyrazol-3-yl)methyl]-1,2-dihydroquinoxalin-2-one
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]piperidine
(1S,5R)-6-(cyclobutylmethyl)-3-[4-(1H-pyrazol-4-yl)butanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2H-1,2,3-benzotriazol-2-yl)-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)acetamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(2,5-difluorophenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
3-[5-(1-methyl-1H-pyrrole-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]pyridine
3-({3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
5-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
2-(1,4-oxazepane-4-carbonyl)-N-(pyridin-2-ylmethyl)aniline
1-[5-(2H-1,3-benzodioxol-4-ylmethyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
7-(2-hydroxyethyl)-2-[2-(6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylphenyl)piperazin-2-one
3-(4-methoxyphenyl)-3-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propan-1-ol
8-(5-phenoxyfuran-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-[3-(hydroxymethyl)phenyl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
8-(2-methoxypropanoyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
4-(cyclopropylmethyl)-1-[(2,3-difluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-[1-(2-methoxypyridine-4-carbonyl)pyrrolidin-2-yl]-1-methyl-1H-1,3-benzodiazole