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3,6-dimethyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
3-(2-fluorophenoxy)-N-[3-(piperidin-1-ylmethyl)phenyl]azetidine-1-carboxamide
N-(1-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
[(3R,4R)-1-(5-phenyl-1,2-oxazole-4-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-(5-oxo-1-phenylpyrrolidin-3-yl)-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
1-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-[(3-methylphenyl)methyl]pyrrolidin-2-one
2-amino-6-(4-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperazin-1-yl)-3,4-dihydropyrimidin-4-one
N-[(2R,3R)-1'-{[3-(2-hydroxyethoxy)phenyl]methyl}-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxyacetamide
2-(2,5-dimethylphenoxy)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]propanamide
1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)-2-[methyl(1-methylpiperidin-4-yl)amino]ethan-1-one
1,3-dimethyl-6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[4-(cyclohex-3-en-1-ylmethyl)piperazin-1-yl]-1-(piperidin-1-yl)ethan-1-one
N-(2-phenylethyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
1-(2-methoxyphenyl)-4-[4-(thiophen-2-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
1-[3-(4-methylphenyl)propanoyl]-4-propyl-1,4-diazepan-5-one
methyl 4-{[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]carbamoyl}butanoate
2-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-(cyclohex-1-en-1-yl)-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
(3S,4S)-4-(dimethylamino)-1-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-ol
(furan-2-ylmethyl)({[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(prop-2-yn-1-yl)amine
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
1-[2-(oxan-2-yl)ethyl]-2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazole
methyl (2S,4R)-4-(2-cyclopropylquinoline-4-amido)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
N-ethyl-N-(4-hydroxybutyl)-3-[(thiophen-2-ylmethyl)amino]benzamide
1-(3-propoxypiperidin-1-yl)-2-(thiophen-3-yl)ethan-1-one
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
1-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-[(3,5-difluorophenyl)methyl]-8-[(4-methoxypyridin-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
7-(2-methoxyethyl)-2-(2-methyl-1,3-benzoxazole-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
dimethyl(3-{2-[1-(2-methylpyridin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-methyl-3-phenylpiperidine
(2S,4R)-1-[2-(2,4-dichlorophenoxy)acetyl]-4-(dimethylamino)pyrrolidine-2-carboxylic acid
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
N-[2-(dimethylamino)ethyl]-3,3,3-trifluoro-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)propanamide
methyl 6-[({[4-(methylsulfanyl)phenyl]methyl}(propyl)amino)methyl]pyridine-2-carboxylate
2-[1-benzyl-4-(2-phenylethyl)piperazin-2-yl]ethan-1-ol
methyl (2S,4R)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(2-methylquinoline-4-amido)pyrrolidine-2-carboxylate
3-[2-(3,4-dimethoxyphenyl)-1H-imidazol-1-yl]propanamide
1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}pent-4-en-1-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(morpholin-4-yl)ethyl]acetamide
N,3,6-trimethyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1-benzofuran-2-carboxamide
4-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-tert-butyl-5-(4-cyclopentylpiperazine-1-carbonyl)-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
4-(1H-imidazol-1-yl)-N-[2-(1H-imidazol-4-yl)ethyl]benzamide
2-({[1-(2H-1,3-benzodioxol-5-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-5-methyl-1,3,4-thiadiazole
N5-[(2-chlorophenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
ethyl 1-[5-(naphthalen-1-yl)-1,2,4-triazin-3-yl]piperidine-3-carboxylate
5-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
N-(2,4-dimethoxyphenyl)-3-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]propanamide