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1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-2,4-dimethyl-1,3-thiazole-5-carboxamide
5-{[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]methyl}-N-ethylpyrimidin-2-amine
2-{4-[4-(benzylamino)piperidin-1-yl]phenyl}-1-(pyrrolidin-1-yl)ethan-1-one
N-(2-methylpropyl)-1-{1-[(2,3,4-trimethoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1,2,3-thiadiazole-4-carboxamide
N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
1-[2-(dimethylamino)-6-(pyridin-4-ylmethyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-4-(pyridin-2-yl)pyrimidin-2-amine
4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1R,9aR)-1-(3-methoxy-2-methylphenoxymethyl)-octahydro-1H-quinolizine
(3S,5R)-N3-cyclohexyl-N5-(2,3-dihydro-1H-inden-5-yl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
1-{5-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]thiophen-2-yl}ethan-1-one
2-methyl-6-[2-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]-2,3-dihydropyridazin-3-one
N-(4-ethoxy-2-fluorophenyl)-7-methyl-12-oxo-3,7,11-triazaspiro[5.6]dodecane-3-carboxamide
2-[2-(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)-2-oxoethyl]-2,3-dihydro-1H-indazol-3-one
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(pyrazine-2-carbonyl)piperidine-2-carboxamide
N-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methylbenzamide
N2,N2,6-trimethyl-N4-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyrimidine-2,4-diamine
(3S,4R)-4-(3-methoxyphenyl)-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]pyrrolidine-3-carboxylic acid
6-[(4-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidin-1-yl)methyl]quinoxaline
methyl 5-[3-(3-methylphenyl)piperidin-1-yl]-5-oxopentanoate
9-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-[4-(pyridin-2-ylmethoxy)phenyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(1R,7S)-3-(2,2-dimethylpropyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-(benzenesulfonyl)-1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]propan-1-one
N-{[1-(2-methoxyphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
1-(2,3-dihydro-1H-indene-1-carbonyl)-4-(thian-4-yl)piperazine
2-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
4-(1-{3-[(1-methylpiperidin-4-yl)oxy]propyl}-4-phenyl-1H-imidazol-5-yl)pyridine
1-[2-(2,2-diphenylethyl)morpholin-4-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-6-methylpyridine
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
N,N-dimethyl-6-(3-{1-[2-(morpholin-4-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyrimidin-4-amine
3-ethyl-8-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N,N-diethyl-1-{1-[(4-ethylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
1-{1-[(5-ethylfuran-2-yl)methyl]pyrrolidin-3-yl}piperidine
4-benzyl-3-ethyl-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1,4-diazepan-5-one
1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-8-(4,4,4-trifluorobutan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-6-(cyclobutylmethyl)-3-(2-phenylacetyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-1-ethyl-6-methyl-1,2-dihydropyridin-2-one
3-{2-[({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)amino]ethyl}-1,3-oxazolidin-2-one
(7S,9aR)-N-cyclohexyl-8-methyl-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
methyl 5-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-2-hydroxybenzoate
3-({[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
(2S,4R)-N-ethyl-1-(naphthalen-2-ylmethyl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
7-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2-oxa-7-azaspiro[4.5]decane
N-[4-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-2-(pyridin-3-yl)acetamide
N-[3-(4-fluorophenyl)phenyl]-1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidine-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(2-methyl-1H-imidazol-1-yl)propanamide