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1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methyl-1,4-dihydroquinolin-4-one
4-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-6-(methoxymethyl)pyrimidine
1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-2-methyl-1,4-diazepan-5-one
3-{[(3R,4S)-3-(2-carboxyethyl)-4-(dimethylamino)piperidin-1-yl]sulfonyl}benzoic acid
5,7-dimethyl-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}pyrido[2,3-d]pyrimidin-4-amine
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
2-{4-[(2,4-dimethoxyphenyl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
(4aS,7aR)-1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
2-[4-(3-chloropyridine-4-carbonyl)-1-(furan-2-ylmethyl)piperazin-2-yl]ethan-1-ol
(3R,4S)-1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-3,4-dimethylpiperidin-4-ol
5-(3,4-difluorophenoxymethyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-methoxyacetamide
N-({7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
N-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}methyl)-3-methylpyridine-2-carboxamide
1-cyclobutanecarbonyl-4-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-1,4-diazepane
1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N,N-bis(prop-2-en-1-yl)piperidine-4-carboxamide
N-[3-(pyridin-2-yl)propyl]-6-({5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}amino)pyridine-3-carboxamide
1-(4-ethylpiperazin-1-yl)-3-[3-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-(1-methyl-1H-imidazol-2-yl)piperidine
9-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-1-phenylcyclohexane-1-carboxamide
3-[3-(dimethylamino)propyl]-5-[(3-fluorophenyl)methyl]-5-{1-[(2E)-4-methylpent-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
1-methyl-8-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-3-ol
4-[(4-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl]piperazine-1-sulfonamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(2-oxopyrrolidin-1-yl)propanamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}acetamide
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)pyridine-2-carboxamide
2-cyclopropyl-9-(2-methoxyacetyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
3-[1-(2-fluorobenzoyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
5-(dimethylamino)-2-{2-[3-(2-ethylphenoxy)azetidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
3-{[5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-phenyl-4H-1,2,4-triazole
(3R,5S)-5-{4-[(2-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}pyrrolidin-3-ol
3-(2,6-dimethoxypyridin-3-yl)-1-{2-[(3-methylpyridin-2-yl)amino]ethyl}urea
1-[2-(cyclohex-1-en-1-yl)ethyl]-1-(cyclopropylmethyl)-3-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-phenoxyethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
6-methyl-4-[3-(1H-pyrazol-1-yl)phenyl]-2,3-dihydropyridazin-3-one
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]acetamide
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-phenylprop-2-ynamide
4-[(1-methyl-1H-pyrazol-4-yl)methyl]-11-({[3-(trifluoromethoxy)phenyl]methyl}amino)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-benzyl-3-[(2,2-dimethylmorpholin-4-yl)methyl]-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
{5-[1-(2,3-dihydro-1H-inden-5-yl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methanol
4-[(4-methoxy-3-methylphenyl)methyl]-3-{2-oxo-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethyl}piperazin-2-one
1-[(1R,2R)-2-phenylcyclopropanecarbonyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[(1-cyclopentylpiperidin-4-yl)methyl]-1-methyl-N-(pyridin-3-ylmethyl)-1H-pyrrole-2-carboxamide