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4-(2,4-difluorobenzoyl)-7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-benzyl-3-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide
(3S,4R)-1-[3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
2,5-dioxo-6-[2-phenyl-2-(piperidin-1-yl)ethyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-(2-aminoethyl)-N,5,6-trimethyl-N-(2-phenylethyl)thieno[2,3-d]pyrimidin-4-amine
3-chloro-4-fluoro-N-[(3R,4R)-4-hydroxypiperidin-3-yl]-1-benzothiophene-2-carboxamide
(2S,4R)-4-(dimethylamino)-1-(5-fluoro-2-methylbenzenesulfonyl)pyrrolidine-2-carboxylic acid
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)furan-3-carboxamide
(4aR,7aS)-1-[2-(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4,6-dimethyl-3-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1H-indol-2-one
1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-4-[(3-methylphenyl)methyl]-1,4-diazepan-5-one
3-cyclopropyl-5-(5-ethoxyfuran-2-yl)-1H-1,2,4-triazole
(3R,4R)-1-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(azepan-1-yl)piperidin-3-ol
4-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1λ6-thiane-1,1-dione
6-[2-(trifluoromethyl)morpholin-4-yl]pyridine-2-carbonitrile
4-benzyl-3-ethyl-1-(1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1,4-diazepan-5-one
4-(5-fluoro-4-methoxypyrimidin-2-yl)benzamide
(1-benzothiophen-2-ylmethyl)({[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
4-(5-methylpyridin-2-yl)-1-[2-(morpholin-4-yl)pyridine-3-carbonyl]piperidin-4-ol
4-[5-(oxolan-3-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]benzene-1-sulfonamide
1,3-dimethyl-4-[2-(2-methylpyrimidin-5-yl)quinoline-4-carbonyl]piperazin-2-one
5-methyl-4-[(pyridin-2-ylmethyl)amino]-N-[2-(thiophen-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-(2-fluoroethyl)-3-{[2-(hydroxymethyl)piperidin-1-yl]sulfonyl}benzamide
8-chloro-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(furan-2-yl)-N-methylquinoline-4-carboxamide
N-[2-(3-fluorophenyl)ethyl]-2-(4-{4-[4-(2-hydroxyethyl)piperazin-1-yl]piperidin-1-yl}phenyl)acetamide
methyl 2-(2-{1-methyl-3-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenoxy)acetate
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1-phenyl-1H-1,2,3-triazole
N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}-2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamide
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[2-(4-chlorophenyl)ethyl]-2-{[2-(pyridin-2-yl)ethyl]amino}acetamide
(2S,4R)-1-cyclopropanecarbonyl-N-ethyl-4-[2-(pyridin-2-ylsulfanyl)acetamido]pyrrolidine-2-carboxamide
[5-({[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]amino}methyl)furan-2-yl]methanol
N-(2,6-dimethoxypyridin-3-yl)-4-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}benzamide
N-[(2-chlorophenyl)methyl]-3-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-yl)propanamide
(3aS,6aS)-1-oxo-2-propyl-5-[3-(thiophen-3-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3,7-dimethyl-11-(5-phenyl-1H-pyrrole-2-carbonyl)-3,7,11-triazaspiro[5.6]dodecane
1-(2-phenylphenyl)-4-(1H-pyrrole-2-carbonyl)piperazin-2-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
2-(8-methoxy-4-methylquinolin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
dimethyl[(5-{[3-(trifluoromethoxy)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]amine
N-[(1,4-dimethylpiperazin-2-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
6-(morpholin-4-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
1-[(4-{[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
4-{[(3-hydroxypropyl)[(5-methylthiophen-2-yl)methyl]amino]methyl}benzonitrile
3-cyclopentyl-5-[(4-fluorophenyl)methyl]-5-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
5-(2-fluorophenyl)-N-(2-methanesulfonylethyl)pyrazolo[1,5-a]pyrimidin-7-amine