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8-(1H-imidazol-4-ylmethyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 4-[benzyl(3-hydroxy-2-methylpropyl)carbamoyl]butanoate
3-[4-(3-hydroxyphenyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
(3S,9aR)-3-[(benzyloxy)methyl]-8-(3,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)pyrimidin-2-amine
4-(naphthalen-2-yloxy)-1-(pyridin-4-ylmethyl)piperidine-4-carboxylic acid
2-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
ethyl 1-{[1-(carbamoylmethyl)-1H-indol-3-yl]methyl}-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
6-[(3R,4R)-4-amino-3-hydroxypiperidine-1-carbonyl]-5-hydroxy-2-(4-methylphenyl)-2,3-dihydropyridazin-3-one
6-{[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
3-chloro-2-fluoro-N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
3-[(3-chlorophenyl)methyl]-1-(pyridin-3-ylmethyl)piperidine-3-carboxylic acid
ethyl 4-[(2-chlorophenyl)methyl]-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
N-[7-oxo-5-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]propanamide
1-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-4-(hydroxymethyl)piperidin-4-ol
9-[5-(ethylsulfanyl)thiophene-2-carbonyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyrrolidin-3-yl)benzamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-(1-methylcyclopropyl)propanamide
3-butyl-4-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-1-methylpiperazin-2-one
4-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]thiomorpholine
3-(3-hydroxyquinoxalin-2-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]propanamide
N-[(3R,4S)-4-cyclopropyl-1-(2,6-diaminopyrimidin-4-yl)pyrrolidin-3-yl]-2-(pyrrolidin-1-yl)acetamide
[(2S,6S)-4-[2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)pyrrolidin-3-ol
2-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
methyl({[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl})[1-(1,2-oxazol-3-yl)ethyl]amine
3-({4-benzyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-2-methoxypyridine
N-[2-(dimethylamino)ethyl]-3-(2-methoxyphenyl)-N-{[7-(methylsulfanyl)-2-(thiophen-2-yl)quinolin-3-yl]methyl}propanamide
2-ethyl-5-(2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)-6-methyl-3,4-dihydropyrimidin-4-one
2-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-6-fluoroquinolin-4-ol
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(4-methoxyphenyl)ethyl]acetamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}oxane-2-carboxamide
2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
3-[4-(2-phenylethyl)piperidine-1-carbonyl]piperidine-1-carboxamide
(2S)-2-{[6-(aminomethyl)-2-methylpyrimidin-4-yl]amino}-4-(methylsulfanyl)butan-1-ol
2-[3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(2-phenylethyl)acetamide
2-fluoro-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-5-sulfamoylbenzamide
2-[1-(3-methylbutyl)-4-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl]ethan-1-ol
1-[1-(cyclohexylmethyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-4-carboxamide
6-({[(1,5-dimethyl-1H-indazol-3-yl)methyl]amino}methyl)-1,4-oxazepan-6-ol
4-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,6-dimethylpyrimidine
9-(cyclopropylmethyl)-1-methyl-4-[(4-methyl-1,3-thiazol-5-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(2,5-difluorobenzoyl)-1-[(5-methylfuran-2-yl)methyl]piperidine
3-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1-(3-methoxy-4-methylphenyl)urea
5-{[(1R,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2,1,3-benzothiadiazole
N-[2-(dimethylamino)ethyl]-3-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}propanamide
1-(carbamoylmethyl)-N-[1-(1H-indol-2-yl)ethyl]-N-methylpiperidine-4-carboxamide
1-cyclohexyl-3-(cyclopropylmethyl)-N-methyl-2-oxo-N-(1H-pyrazol-3-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-(benzenesulfonyl)-N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
2-{2-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyrazine