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6-cyclopentyl-N,1-dimethyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}propanamide
2,6-dimethyl-5-(2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one
N-methyl-3-(propan-2-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-3-(2-oxopyrrolidin-1-yl)propanamide
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(oxan-2-ylmethyl)amine
[(3aS,6aS)-2-[2-(ethylamino)pyrimidine-5-carbonyl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
[5-({3-[(4-fluorophenyl)amino]piperidin-1-yl}methyl)-2-(propan-2-yloxy)phenyl]methanol
5-methyl-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}imidazo[1,2-a]pyridine-2-carboxamide
2-(2,5-dimethoxyphenyl)-N-[1-(4-methyl-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]acetamide
7-[2-(4-chlorophenyl)morpholine-4-carbonyl]-1H-indole
methyl (2S,4R)-4-hydroxy-1-{[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}pyrrolidine-2-carboxylate
1-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
(1R,5R)-6-(5-acetylthiophene-2-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
(1R,2S)-N-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-2-phenylcyclohexan-1-amine
2-ethyl-4-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}pyrimidine
(3S,4S)-1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
2-(1,4-dimethylpiperazin-2-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(4-fluorophenyl)-1-(1-propylpiperidin-4-yl)piperidin-3-amine
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrimidin-2-amine
(2S,4S,5R)-4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-methyl-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
N-[1-(7-{[4-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-3-methylbutyl]-2-methoxyacetamide
6-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-1,2-dihydropyridin-2-one
1-[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]-2-phenylethan-1-ol
2-(2-fluorophenoxymethyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1,3-oxazole-4-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]propan-1-one
4-(4-chlorophenyl)-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methylbutanamide
N,N-dimethyl-7-(1-methyl-1H-imidazole-5-carbonyl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-4-oxo-N-(pyridin-2-ylmethyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
4-{7-[3-(trifluoromethyl)benzoyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}morpholine
N-(2-{7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
1-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-(dimethylamino)-2-(3-fluorophenyl)-N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)acetamide
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]cyclobutanecarboxamide
1-(3-methoxyphenyl)-4-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
3-cyclopropyl-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
1-{5-[(2-propyl-2,5-dihydro-1H-pyrrol-1-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidine
1-(4-{4-[4-(pyridin-3-yl)pyrimidin-2-yl]piperazin-1-yl}phenyl)ethan-1-one
1-(dimethyl-1,3-thiazole-5-carbonyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
7-fluoro-1-methyl-2-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
methyl (2S,4S)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]-1-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
3-[2-(3-fluorophenyl)ethyl]-1-[5-(methoxymethyl)furan-2-carbonyl]piperidine
6-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
3-{2-[3-(2-chlorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione