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1-[6-methyl-2-(methylamino)pyrimidin-4-yl]-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidine
1-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
5-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one
[(5-{1-[(2,6-difluorophenyl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
7-fluoro-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-methylquinoline-4-carboxamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
3-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-1-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)urea
1-(3,4-dimethylphenyl)-N-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
methyl 3-[(2,3-difluorophenyl)methyl]-9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
8-(1H-indol-2-ylmethyl)-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(butan-2-yl)-3-fluoro-2-methoxy-N-(pyridin-3-ylmethyl)benzamide
3-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-4H-chromen-4-one
4-(3-benzyl-1H-pyrazol-5-yl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
(3aR,6aR)-2-acetyl-5-[3-(benzyloxy)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-[2-(2-methoxyphenyl)ethyl]acetamide
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[2-(1H-imidazol-1-yl)ethyl]methylamine
N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]-3-(3,4-difluorophenyl)propanamide
5-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-3-(thiophen-2-ylmethyl)-1,2,4-oxadiazole
2-(1,5-dimethyl-1H-indazol-3-yl)benzamide
(1R,4S)-2-{2-[(E)-2-phenylethenyl]pyridine-3-carbonyl}-2-azabicyclo[2.2.1]heptane
4-[(2-chlorophenyl)methyl]-1-(thiophen-2-ylmethyl)-1,4-diazepan-5-one
2-(2-methyl-6-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}pyrimidin-4-yl)ethan-1-amine
1-(5-hydroxypyrazine-2-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
5-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)-2,1,3-benzothiadiazole
6-(4-chlorophenyl)-N-[2-(oxolan-3-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl](ethyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]amine
N4-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-[1-(1-{spiro[2.5]octane-1-carbonyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-ol
6-methoxy-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(2R,3R)-3-(1H-imidazol-1-yl)-1'-[(2-methyl-1,3-thiazol-5-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
7-(cyclopropylmethyl)-2-(3,4,7-trimethyl-1H-indole-2-carbonyl)-2,7-diazaspiro[4.5]decane
methyl 4-({1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidin-4-yl}formamido)butanoate
2-cyclohexyl-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1,3-benzoxazole-6-carboxamide
2-{3-[(4-fluorophenyl)methoxy]azetidine-1-carbonyl}-3,5-dimethyl-1H-indole
2-(hydroxymethyl)-N-[3-(prop-2-en-1-yloxy)phenyl]azepane-1-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2-(2-ethyl-1H-1,3-benzodiazol-1-yl)butanamide
methyl 6-[(3-chloro-4-hydroxyphenyl)methyl]-2-[methyl(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[2-(pyridin-3-yloxy)propyl]amine
[(6-methoxy-2H-chromen-3-yl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
methyl 3-(2-methoxyacetamido)-5-{[(4-methoxyphenyl)methyl]amino}-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[3-(3,4-difluorophenyl)-1H-pyrazol-1-yl]-N-(1,3-dimethyl-1H-pyrazol-5-yl)acetamide
1-{1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-oxopropan-2-yl}pyrrolidin-2-one
4-benzyl-3-ethyl-1-(1-methyl-1H-pyrazole-3-carbonyl)-1,4-diazepan-5-one
2-(2-{1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
1,6-dimethyl-3-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
11-{[(2,6-difluorophenyl)methyl]amino}-4-[3-(propan-2-yloxy)propyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-methyl-2-(pyridin-4-yl)-N-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine