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2-[2-(methylamino)-1,3-thiazole-4-carbonyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(morpholin-4-yl)-6-[3-(morpholin-4-ylmethyl)phenyl]pyrimidin-4-amine
6-ethyl-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]pyrimidin-4-amine
N-[2-(4-{[ethyl(methyl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]methanesulfonamide
N-[3-(1H-imidazol-1-yl)propyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
methyl 7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-3-(4-phenylbutanoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
1-(6-chloro-1,3-benzothiazol-2-yl)-N-[(3-methylpyridin-2-yl)methyl]piperidin-4-amine
3-(2-methyl-1H-indol-1-yl)-1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
2-methoxy-1-[1'-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
2-(dimethyl-1,3-thiazol-5-yl)-1-{spiro[indene-1,4'-piperidine]-1'-yl}ethan-1-one
N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-4-methoxy-N-(2-methoxyethyl)benzamide
(3R,4R)-3-hydroxy-N-[(4-methoxyphenyl)methyl]-4-methyl-3-(propan-2-yl)pyrrolidine-1-carboxamide
1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]-4-(2-methylphenyl)-1,4-diazepane
ethyl 1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
4-{[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]methyl}benzonitrile
methyl (2S,4R)-1-[(2,5-difluorophenyl)methyl]-4-[3-(4-methylphenyl)propanamido]pyrrolidine-2-carboxylate
2-({[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}amino)propan-1-ol
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N,N-dimethyl-2-{N-methyl-1-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}propanamide
methyl 4-[(4-{[3-(furan-2-yl)phenyl]carbamoyl}piperidin-1-yl)methyl]benzoate
N-[3-(dimethylamino)-2,2-dimethylpropyl]-6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
1-benzyl-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
1-[(3S)-1-benzylpyrrolidin-3-yl]-5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazole
N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-(thiophen-2-ylmethyl)piperidine-2-carboxamide
1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidine
N-[4-(4-{[(1-benzyl-1H-pyrazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]pyrazine-2-carboxamide
{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}(furan-2-ylmethyl)(thiophen-3-ylmethyl)amine
4-[(1S,2R)-1-hydroxy-2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]phenol
3-(1H-1,3-benzodiazol-2-ylmethyl)-9-methoxy-7-oxo-N-[3-(1H-pyrazol-1-yl)propyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(5-methyl-1,3-thiazol-2-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
2-(1-methyl-3-oxopiperazin-2-yl)-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
N,N-dimethyl-3-[5-(morpholine-4-carbonyl)pyridin-2-yl]aniline
1-[(2,4-difluorophenyl)methyl]-5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
N-cyclopropyl-3-[5-(1-methyl-1H-pyrrole-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
(cyclopropylmethyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propylamine
N-[(3S,4R)-1-(3-cyano-5-fluorobenzoyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
5-(5-fluoro-1-methyl-1H-indazol-3-yl)-1,2,3,4-tetrahydroisoquinoline
5-({1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-2-(methylsulfanyl)pyrimidine
2-{4-[3-(2-chlorophenyl)propyl]piperazin-1-yl}pyrazine
3-methyl-N-[1-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]butanamide
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
(4aS,7aR)-1-(2-ethoxybenzoyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
N-(pyridin-2-ylmethyl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-ethyl-N-(2-fluorophenyl)-2,5-dihydro-1H-pyrrole-1-carboxamide
2-tert-butyl-4-hydroxy-N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}pyrimidine-5-carboxamide