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2-ethyl-9-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopentyl-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-(3-phenylprop-2-yn-1-yl)propanamide
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
2-[(4aR,7aS)-4-[(2-fluorophenyl)carbamoyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
3-(oxolan-2-ylmethyl)-5-{1-[4-(2-oxopyrrolidin-1-yl)benzoyl]piperidin-4-yl}-5-propylimidazolidine-2,4-dione
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-3-(pyridin-4-yl)propanamide
2-{2,5-dioxo-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl}-N-methyl-N-(quinoxalin-6-ylmethyl)acetamide
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propanamide
2-[5-(2-methylbutyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
2-(2,5-dimethylphenoxy)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}propanamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-7-fluoro-2-methylquinoline
2-[5-(1-ethyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]pyridine
2,3,5,6-tetramethyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)benzamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
[2-ethoxy-5-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenyl]methanol
(3S,4R)-N,N-dimethyl-4-(propan-2-yl)-1-(pyridin-4-ylmethyl)pyrrolidin-3-amine
4-{2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]acetyl}-1-phenylpiperazin-2-one
N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]propanamide
[(3,4-difluorophenyl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
1-[(4-chlorophenyl)methyl]-4-(1,2-oxazolidine-2-carbonyl)-1H-1,2,3-triazole
2-(pyridin-3-yl)-5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]pyrimidin-4-ol
N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]cyclobutanecarboxamide
(1S,5R)-6-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
5-methoxy-2-{[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-4H-pyran-4-one
methyl 1-(1-{4-[2-(3-fluorophenyl)acetamido]phenyl}piperidin-4-yl)piperidine-4-carboxylate
2-(2-chlorophenyl)-3-methyl-N-[(3-methylpyridin-2-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-{2-[methyl(2-methylpropyl)amino]ethyl}-8-(1-methyl-1H-pyrazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(5-chloro-2-fluorobenzoyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-methyl-1-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]urea
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
methyl 5-{[(2-chloro-3,4-dimethoxyphenyl)methyl]amino}-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
9-methoxy-3-[(3-methylquinoxalin-2-yl)methyl]-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
methyl 6-[(2-methylphenyl)methyl]-2-(morpholine-4-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-{[(6-chloropyridin-3-yl)methyl](pyridin-2-ylmethyl)amino}-2-methylpropan-1-ol
3-(2-methoxyethyl)-1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}piperidine-3-carboxylic acid
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)pyrrolidin-3-yl]acetamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-(1-ethyl-3-oxopiperazin-2-yl)acetamide
2-{4-[(4,8-dimethoxynaphthalen-1-yl)methyl]piperazin-1-yl}acetic acid
3-{1-[5-(3-fluorophenoxymethyl)-1H-pyrazol-3-yl]-N-methylformamido}propanamide
ethyl 4-benzyl-1-{[3-(ethoxycarbonyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylate
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
ethyl N-({1-[(3R,5S)-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazol-4-yl}methyl)-N-methylcarbamate
{4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]morpholin-2-yl}methanamine
2-[3-(morpholin-4-ylmethyl)phenyl]pyridine-3-carbonitrile
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-5-phenyl-1,2-oxazole
9-[(2R)-2-amino-3-phenylpropanoyl]-2-(cyclopropylmethyl)-2,9-diazaspiro[5.5]undecan-3-one