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(1-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}piperidin-4-yl)methanol
7-methyl-2-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
5-chloro-N-[1-(cyclohexylmethyl)piperidin-3-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-diethylacetamide
2-[1-({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)piperidin-4-yl]ethan-1-ol
1'-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-[(4,6-dimethylquinolin-2-yl)sulfanyl]-1-(6-hydroxy-1,4-oxazepan-4-yl)propan-1-one
methyl (2S,4R)-1-{3-[(4-fluorophenyl)formamido]propanoyl}-4-hydroxypyrrolidine-2-carboxylate
2-(1H-imidazol-2-yl)-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}benzamide
4-[2-ethyl-7-(furan-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1,4-oxazepane
N-methyl-2-[4-(3-{[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl}propanoyl)morpholin-3-yl]acetamide
{4-[1-benzyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]phenyl}methanamine
2-(carbamoylamino)-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]acetamide
2-(dimethylamino)-N-{[1-(ethoxymethyl)cyclobutyl]methyl}-2-(2-methylphenyl)acetamide
{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]methylamine
(3aS,6aS)-2-ethyl-5-[3-(1,2-oxazinan-2-yl)propanoyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-cyclopropyl-5-(1,3-dimethyl-1H-pyrazol-4-yl)-1-(2-phenylethyl)-1H-1,2,4-triazole
1-[4-({4-[4-(methylsulfanyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
methyl (2R,4S)-4-hydroxy-1-(2-phenylacetyl)piperidine-2-carboxylate
methyl 7-oxo-9-[2-(pyridin-2-yl)ethoxy]-3-[4-(thiophen-2-yl)butanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2R,3S,6R)-3-phenyl-5-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
(1S,4S)-2-{5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carbonyl}-2-azabicyclo[2.2.1]heptane
8-methoxy-N-[(5-methylpyrazin-2-yl)methyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
6-[2-(2-methoxyethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-(furan-2-ylmethyl)-2,3-dimethoxy-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}benzamide
[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
(3S,4R)-3-benzyl-N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1-methylpiperidin-4-amine
N,N-diethyl-1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-3-carboxamide
7-(2-methoxyphenyl)-2-[3-(pyrrolidin-1-yl)propyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
7-fluoro-4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-2-methylquinoline
3-{1-[3-(3-chlorophenyl)propanoyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
(1R,5R)-6-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[(2R)-1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-1-oxopropan-2-yl]acetamide
2-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]pyridine
4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-(piperidin-1-yl)pyrimidine
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
1-(adamantan-2-yl)-4-[(2S,4S)-4-[(4-methoxyphenyl)sulfanyl]-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carbonyl]piperazine
1-(4,7-dimethylquinazolin-2-yl)-N-(2-methylpropyl)azepan-4-amine
2-methyl-N-({3-methyl-7-[2-(2,3,6-trifluorophenyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-3-carboxamide
3-[(4-{4-[ethyl(methyl)amino]pyrimidin-2-yl}piperazin-1-yl)methyl]benzonitrile
2-{4-[(2-ethyl-4-methyl-3-oxopiperazin-1-yl)methyl]-2-methoxyphenoxy}acetamide
6-oxo-1-(2-phenylethyl)piperidine-3-carboxylic acid
{2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}urea
(3S,4R)-1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
4-{[1-(4-fluorophenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-2,3-dihydro-1H-pyrazol-3-one
1-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-3-phenylpiperazine
4-[(1-acetylpiperidin-4-yl)oxy]-3-chloro-N-cyclopentylbenzamide
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide