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5-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-N-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
5-{3-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-oxopropyl}-5-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-2-one
3-{2-[4-(4-acetylphenyl)piperazin-1-yl]-2-oxoethyl}-1-(3-methoxypropyl)-3-phenylpyrrolidine-2,5-dione
[(3R,4R)-1-(4-cyclopentylpyrimidin-2-yl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-(oxolan-2-ylmethyl)piperazine
9-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-hydroxy-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
N-methyl-N-[2-(2-methylphenyl)-1-[1-(quinoline-2-carbonyl)piperidin-4-yl]ethyl]-2-(1H-pyrazol-1-yl)acetamide
N-{[6-(3-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(2-methoxyethyl)-1,3-thiazole-5-carboxamide
N-cyclopentyl-2-({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)propanamide
8-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-methyl-4-(2-methylpropyl)-N-[4-(methylsulfanyl)phenyl]-3-oxopiperazine-1-carboxamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-benzyl-N-ethyl-1-[(1-ethylpiperidin-3-yl)methyl]piperidin-4-amine
4-[(1S,2S)-2-hydroxycyclohexyl]-N-[2-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperazine-1-carboxamide
4-[(2-methoxyethyl)amino]-5-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
3,5-dimethyl-1-[(4-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}phenyl)methyl]-1H-pyrazole
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidine
(4aS,8aR)-1-(pyridin-2-ylmethyl)-6-(pyrimidin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
3-[(1-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-3-yl)methyl]benzoic acid
1-(1,2,3,4-tetrahydroquinolin-1-yl)-3-[2-(trifluoromethyl)morpholin-4-yl]propan-1-one
4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-methyl-2-(propan-2-yl)pyrimidine
2-amino-4-(1,5-dimethyl-1H-pyrazol-4-yl)-6-{4-[(dimethylamino)methyl]thiophen-2-yl}pyridine-3-carbonitrile
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-6-methylpyridazin-3-amine
3-{1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-1,3-oxazolidin-2-one
(2S,4S)-N-ethyl-4-(furan-3-amido)-1-[2-(thiophen-2-yl)acetyl]pyrrolidine-2-carboxamide
(1R,3s,6r,8S)-4-{5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carbonyl}-4-azatricyclo[4.3.1.13,8]undecane
4-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
methyl 4-{[(2-{1-[(5-chlorothiophen-2-yl)methyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
4-ethyl-3-{1-[(2S)-2-phenylbutanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1H-1,2,3-triazole
3-[1-(2H-1,3-benzodioxol-5-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]pyridin-2-ol
1-{3-[(1-methylpiperidin-4-yl)methyl]-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl}cyclopropane-1-carboxamide
4-{[3-(5-fluoropyridin-2-yl)phenyl]methyl}morpholine
1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-(3-methylpyridin-2-yl)piperazine
4-[(1-acetylpiperidin-4-yl)oxy]-N-[(5-fluoro-2-methylphenyl)methyl]-3-methoxybenzamide
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]pyridine
2-(ethylsulfanyl)-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
2-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}pyrrolidin-2-yl)pyridine
N-[3-(aminomethyl)phenyl]-4-(furan-2-carbonyl)-1,4-diazepane-1-carboxamide
N-[1-(hydroxymethyl)cyclopentyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-benzyl-N-ethylacetamide
2-[5-(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)-3-phenyl-1H-1,2,4-triazol-1-yl]-3-methylpyridine
(5S,9aS,9bS)-2-cyclopentyl-5-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-methyl-4-phenylpyrimidine-5-carboxamide
[(3R,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methanol
methyl (2S)-2-({5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazol-3-yl}formamido)-4-methylpentanoate
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-7-oxo-3-(oxolane-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{4-[(4-methoxy-2,3-dimethylphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol