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1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydroquinolin-2-one
3-chloro-N-(4-{4-[(3-ethoxypropyl)amino]piperidin-1-yl}phenyl)benzamide
(3S)-1-[(5-chlorothiophen-2-yl)methyl]-N,N-dimethylazepan-3-amine
(3S)-3-benzyl-4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-one
3-(oxolan-3-yl)-5-(4-propylphenyl)-1,2,4-oxadiazole
1-[(1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
methyl 7-oxo-3-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(3S,4S)-1-(1H-imidazol-2-ylmethyl)-4-[4-(morpholine-4-carbonyl)piperazin-1-yl]pyrrolidin-3-ol
ethyl 5-(2-methoxyacetyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
5-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,2,3-benzotriazole
4-[4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-6-(1H-pyrazol-1-yl)pyrimidine
N-cyclopropyl-1-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
3-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
(3R,4R)-1-[(4,5-dimethylfuran-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
4-{5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl}benzamide
2-(3-cyclohexylpropanamido)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
4-(pyrrolidin-1-yl)-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(4-methylbenzoyl)pyrrolidin-3-yl]methanol
1-(5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-1H-pyrazole-4-carbonyl)-N,N-diethylpyrrolidin-3-amine
4-{[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]amino}-1-phenylpyrrolidin-2-one
2-(5-acetyl-4-methylpyrimidin-2-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-benzyl-5-methyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-2-(dimethylamino)-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethan-1-one
(1S,5R)-3-[(3-chloro-4-methoxyphenyl)methyl]-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(2-methoxyphenoxy)-1-(pyridin-2-yl)piperidine-4-carboxylic acid
7-fluoro-3-methyl-2-[2-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1H-indole
(3S,4R)-4-(3-methoxyphenyl)-1-(4,4,4-trifluorobutanoyl)pyrrolidine-3-carboxylic acid
N-cyclopentyl-3-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]propanamide
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]pyridin-2-amine
(3S,4R)-1-[3-(dimethylamino)benzoyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-[(3R,5S)-1-butyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
(1R,5R)-6-benzyl-N-(3-methoxyphenyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
8-(cyclohex-3-en-1-ylmethyl)-1-ethyl-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-butyl-1H-imidazol-4-yl)-1-(3-methoxypropyl)-1H-imidazole
(2,1,3-benzoxadiazol-5-ylmethyl)({[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-[1-(4-chlorophenyl)ethyl]-1-(4,7-dimethylquinazolin-2-yl)piperidine-4-carboxamide
2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-2-phenoxybutanamide
1-{[2-(furan-2-yl)phenyl]methyl}-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
2-(dimethylamino)-2-(4-fluorophenyl)-N-[3-(methylsulfanyl)propyl]acetamide
9-(5-ethyl-2-methylpyrimidin-4-yl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1,3-dimethyl-4-(2-phenylbenzoyl)piperazin-2-one
methyl({[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl})[1-(1,3-thiazol-2-yl)ethyl]amine
(3R,4R)-1-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
2-ethyl-6-methyl-N-[3-(morpholin-4-yl)propyl]-4-oxo-1-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-(4-hydroxyphenyl)-N-(1-methoxybutan-2-yl)-1H-pyrazole-5-carboxamide
2-(4-methyl-6-{4-[(oxolan-3-ylmethyl)amino]piperidin-1-yl}pyrimidin-2-yl)phenol
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-3,3,3-trifluoropropanamide
5-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
N-methyl-N-[2-(phenylsulfanyl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine