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N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-5-methyl-N-[(3S)-2-oxoazepan-3-yl]thiophene-2-carboxamide
1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]-3-propoxypiperidine
2-{[(4-fluorophenyl)methyl][(6-methylpyridin-2-yl)methyl]amino}butan-1-ol
3-{1-[(4-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-1-[2-(morpholin-4-yl)ethyl]urea
N-[2-(pyrrolidin-1-yl)ethyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-benzyl-N-[(1-ethylpyrrolidin-2-yl)methyl]-2-methyl-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carboxamide
N-(pyridin-2-ylmethyl)-1-{1-[2-(pyridin-4-yl)acetyl]piperidin-4-yl}piperidine-4-carboxamide
2-{[3-(hydroxymethyl)piperidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-(cyclopropylmethyl)-1-(5-ethyl-2-methylpyrimidin-4-yl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-methyl-1,3-thiazole-4-carboxamide
N,N,8-trimethyl-2-[1-(pyridin-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
7-(pyrrolidin-1-ylmethyl)-4-[3-(trifluoromethyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-benzyl-3-{1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]piperidin-4-yl}-N-methylpropanamide
8-[2-(4-methanesulfonylphenyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
6-(2-aminoethyl)-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpyrimidin-4-amine
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
N-(2-methoxyethyl)-N-(propan-2-yl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-[(4-fluorophenyl)methyl]-4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
1-[4-(morpholine-4-carbonyl)phenyl]-N-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-amine
N-[(5-chlorothiophen-2-yl)methyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
N-[2-(pyridin-4-yl)ethyl]-2-[4-(thiophene-3-carbonyl)morpholin-3-yl]acetamide
4-[(4-fluorophenyl)methyl]-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-1,4-diazepan-5-one
3-{[(2S)-2-benzyl-3-oxopiperazin-1-yl]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
methyl (1S,3R,3aR,6aS)-3-[(3Z)-hex-3-en-1-yl]-1-(hydroxymethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2,8-diazaspiro[4.5]decane
4-(3,5-difluoropyridine-2-carbonyl)-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
4-(5-chloro-2-methylphenyl)-N-(1-methyl-1H-1,3-benzodiazol-6-yl)piperazine-1-carboxamide
(1-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-3-[(2-fluorophenyl)methyl]piperidin-3-yl)methanol
1-[2-(3-hydroxyazetidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
6-[(4-fluoro-3-methoxyphenyl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
7,7-dimethyl-2-[2-(pyridin-3-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-{[4-(1-cyclohexylpyrrolidin-3-yl)piperidin-1-yl]methyl}pyridine
(3R,4S)-4-(3-methoxyphenyl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]pyrrolidin-3-amine
1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-3-(4-phenylbenzoyl)piperidine
2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N,N-diethylacetamide
N-({1-[(2-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)-5-methoxyfuran-2-carboxamide
N-[2-methyl-3-(pyrrolidin-1-yl)phenyl]-4-(6-methylpyridin-2-yl)piperazine-1-carboxamide
(2S,4R)-N-ethyl-1-(furan-3-ylmethyl)-4-[2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetamido]pyrrolidine-2-carboxamide
N,N-dimethyl-1-(2-methylpropyl)-5-{[3-(methylsulfanyl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[(3R,4S)-1-(5-fluoro-2-methoxybenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
(1S,6R)-9-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,3,5-trimethyl-1H-indole-2-carboxamide
1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(4H-1,2,4-triazol-4-yl)propan-1-one
2-methoxy-N-({5-[(5-methylthiophen-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
2-(1-{[1-(furan-2-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
4-(1-methylazepane-2-carbonyl)-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
2-{3-[3-(thiophen-2-yl)-1H-pyrazol-1-yl]phenoxy}acetamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-(pyridine-2-carbonyl)piperazin-2-yl}ethan-1-ol
2-amino-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]-6-(propan-2-yl)-5-propylpyridine-3-carbonitrile