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3-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amino]methyl}phenol
5-cyclopropanecarbonyl-1'-[3-(5-methylfuran-2-yl)butyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(4-ethylpiperazin-1-yl)-3-[3-({[2-(pyridin-3-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-(oxolan-2-ylmethyl)-9-[2-(pyrazin-2-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[1-(2-phenylethyl)-5-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,4-diazepan-5-one
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-N'-(2-methylphenyl)propanediamide
7-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-2-ethyl-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
1-(1H-1,2,3-benzotriazol-4-yl)-3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]urea
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[2-(methylamino)ethyl]pyrimidine-5-carboxamide
[5-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)furan-2-yl]methanol
methyl 4-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-4-oxobutanoate
4-(2-methoxyphenyl)-2-methyl-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperazine
3-(2-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-2-(4-methoxyphenyl)acetamide
N-[2-(4-chlorophenyl)propyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
3-(3-methylbutyl)-8-[3-(1-methylpiperidin-3-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 3-benzamido-1-(oxolan-2-ylmethyl)-5-(propylamino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-({3-hydroxy-1-[(3-methylphenyl)methyl]-2-oxopiperidin-3-yl}methyl)piperazin-2-one
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamide
2-(4-fluorophenyl)-4-(3-propyl-1H-pyrazole-4-carbonyl)morpholine
2-{9-[2-(4-methylphenoxy)acetyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
1-[2-(1H-imidazol-4-yl)ethyl]-2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazole
1-methyl-2-{thieno[3,2-d]pyrimidin-4-ylmethyl}piperidine
2-[(5-{[benzyl(methyl)amino]methyl}-1,2-oxazol-3-yl)formamido]-N-cyclopropylacetamide
(2-{[4-(4-ethenylbenzoyl)piperazin-1-yl]methyl}phenyl)methanol
6-[2-chloro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
1-(4-cyanobenzoyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-(3,5-dimethoxyphenyl)-3-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}urea
2-methyl-N-{[1-(pyridin-3-ylmethyl)piperidin-4-yl]methyl}pyrimidine-5-carboxamide
2,5-dimethyl-3-(4-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrazine
3-methoxy-N-[(3R,4S)-1-[(2E)-2-methylbut-2-en-1-yl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]propanamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[2-(3,4-dimethylphenyl)ethyl]acetamide
4-[2-(2-chlorophenyl)ethyl]-11-{[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(4-methoxyphenyl)-4-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
2-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-1-yl}-2-[4-(propan-2-yloxy)phenyl]acetic acid
N-[(2R,3R)-1'-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
9-ethyl-1-methyl-4-(2-methyl-5-propylpyrimidin-4-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-[ethyl(methyl)amino]acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
(4aS,8aR)-6-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-methyl-N-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]thian-4-amine
ethyl 4-(2-phenylethyl)-1-[3-(pyridin-4-yl)propanoyl]piperidine-4-carboxylate
4-methyl-6-{4-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-1-yl}pyrimidin-2-amine
3-[(3R,4S)-4-(morpholin-4-yl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-yl]propanoic acid
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(2-methoxyphenyl)-2-methylpiperazine
N3-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N5-[2-(pyridin-4-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]azetidine-2-carboxylic acid
(3S,4S)-4-(propan-2-yl)-1-(thiophene-3-carbonyl)pyrrolidine-3-carboxylic acid
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine