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3-(2-oxo-2-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}ethyl)-3,4-dihydroquinazolin-4-one
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-4-(pyridin-3-yl)pyrimidin-2-amine
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]cyclopropanecarboxamide
8-[5-(4-methoxyphenyl)furan-2-carbonyl]-1-oxa-8-azaspiro[4.6]undecane
N-[3-(2-methoxybenzamido)phenyl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
2-(2,4-dichlorophenoxy)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]acetamide
N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-[(2-hydroxyethyl)(methyl)sulfamoyl]benzamide
2-{4-chloro-2-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]phenoxy}acetamide
5-{6-[3-(dimethylamino)propoxy]pyridin-3-yl}-1H-indazol-3-amine
methyl 1-(benzyloxy)-2-oxo-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
4-(3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-2,5-dimethyl-1H-pyrrol-1-yl)-4H-1,2,4-triazole
methyl 3-[4-(3,5-dimethylphenyl)-3-oxopiperazine-1-carbonyl]benzoate
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-5-phenyl-1,2-oxazole-3-carboxamide
2-(dimethylamino)-N-(1-{1-[3-(2-methoxyphenyl)propanoyl]piperidin-4-yl}-2-phenylethyl)-N-methylacetamide
1-[1-ethyl-5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
1-[6-(2-methoxyquinolin-3-yl)pyridin-2-yl]ethan-1-ol
(3R)-1-({1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)pyrrolidin-3-ol
1-methyl-2-oxo-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}-1,2-dihydroquinoline-3-carboxamide
2-methoxy-6-({methyl[1-(pyridin-4-yl)ethyl]amino}methyl)phenol
N,3,5,7-tetramethyl-N-(thian-4-yl)-1H-indole-2-carboxamide
2-(3-hydroxyphenyl)-2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]acetic acid
N-benzyl-5-(4-chloro-2-methoxyphenoxymethyl)-N-(2-hydroxyethyl)-1,2-oxazole-3-carboxamide
N,N-diethyl-8-methyl-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
ethyl 2-{2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-methylacetamido}acetate
3-[(1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)oxy]pyridine
5-methoxy-1-methyl-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1H-indole
1-{2-[4-fluoro-3-(trifluoromethyl)phenyl]pyrimidin-4-yl}piperidin-4-ol
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]pent-4-enamide
3-{[1-(6-ethoxy-4-methylquinazolin-2-yl)piperidin-4-yl]amino}-1λ6-thiolane-1,1-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-9-methoxy-7-oxo-3-[2-(thiophen-2-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-(5-propyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]methanol
1-(2-{methyl[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amino}pyrimidin-4-yl)piperidin-4-ol
1-[(5-chlorofuran-2-yl)methyl]-4-(oxan-4-yl)piperazine
4-(2-{1-[5-(5-methylfuran-2-yl)-1,2,4-triazin-3-yl]piperidin-2-yl}ethyl)phenol
5-ethyl-6-methyl-N4-{3-[(1-methylpiperidin-4-yl)oxy]propyl}pyrimidine-2,4-diamine
(3R,4R)-3,4-dimethyl-1-[2-(methylamino)pyridine-4-carbonyl]pyrrolidin-3-ol
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidin-4-ol
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
4-(3-methylphenoxy)-1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidine-4-carboxylic acid
3-[6-(dimethylamino)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]-1-[1-(pyridin-4-yl)propan-2-yl]urea
3-ethyl-5-{1-[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazole
1-{[1-(methoxymethyl)cyclopentyl]methyl}-5-(1-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazole
(4aS,7aR)-1-(1H-imidazol-2-ylmethyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2,3-dihydro-1H-inden-2-yl)-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N4-[(5-methylpyrazin-2-yl)methyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
6-[3-oxo-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propyl]-2,3,4,5-tetrahydropyridazin-3-one
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
2-(2,4-dichlorophenoxy)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]acetamide
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine