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1-{4-[2-(4-chlorophenyl)morpholin-4-yl]piperidin-1-yl}butan-1-one
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-1-phenylcyclohexane-1-carboxamide
2,6-difluoro-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)benzamide
(3S,4R)-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
5-[(2S)-1-(5-phenyl-1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
4-(naphthalen-1-yl)-3-(1H-pyrazol-4-yl)-4H-1,2,4-triazole
(1S,5R)-6-[2-(benzyloxy)benzoyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
N-[2-(7-{2-[3-(trifluoromethyl)phenyl]acetyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclohexanecarboxamide
6-ethyl-N4-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N4,5-dimethylpyrimidine-2,4-diamine
1-[7-(hydroxymethyl)-9-(pyrimidin-2-yl)-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one
4-(3-fluoro-4-methylbenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[2-(pyridin-3-yloxy)propyl]butanamide
[(2-methyl-1,3-thiazol-4-yl)methyl][4-methyl-4-(methylsulfanyl)pentan-2-yl]amine
4-methoxy-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyridine
6-[4-(hydroxymethyl)piperidin-1-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(4-fluoro-3-methoxyphenyl)methyl]pyrrolidin-3-yl]methanol
7-(3-chlorophenyl)-4-[(3-hydroxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[3-(2,3-dimethoxyphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]thiomorpholine
4-(2,3-dihydro-1H-inden-2-yl)-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(3-benzyl-1H-1,2,4-triazol-5-yl)-4-(pyrimidin-2-yl)piperazine-1-carboxamide
1-[2-(dimethylamino)ethyl]-3-(1-methyl-1H-pyrazol-4-yl)-1-[(5-methylthiophen-2-yl)methyl]urea
2-(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-imidazol-2-yl)pyridine
9-[(4-chloro-2-fluorophenyl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)piperidin-3-yl]methyl}acetamide
N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-1'-(4,4,4-trifluorobutanoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
4-[4-(6-chloropyridin-3-yl)-1H-1,2,3-triazol-1-yl]-1-(2-methoxyethyl)pyrrolidin-2-one
1-(2,3-dihydro-1H-inden-2-yl)-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
7-(3-methanesulfonylbenzoyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(2H-1,3-benzodioxol-5-yl)-2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
2-ethyl-5-{1-[2-(3-methoxyphenyl)ethyl]-1H-imidazol-2-yl}-4-methyl-1H-imidazole
2,2-dimethyl-3-({5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propan-1-ol
N-{2-[4-({[(2-methoxynaphthalen-1-yl)methyl](methyl)amino}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}methanesulfonamide
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-(7-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
3-(3-methylbutyl)-5-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-(piperidin-3-yl)-N-{3-[(pyridin-3-yl)amino]propyl}benzamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(3,4-dimethylphenyl)methyl]piperidin-3-yl}propanamide
1-(3-{[7-acetyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
4-(4-{3-tert-butyl-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)-1,2,3-thiadiazole
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-cyclopentyl-N-propyl-1H-pyrazole-3-carboxamide
methyl (2S,4R)-1-[6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-hydroxypyrrolidine-2-carboxylate
1-methyl-5-[(2S)-2-(morpholine-4-carbonyl)pyrrolidine-1-carbonyl]-1H-1,3-benzodiazole
1-(4-methoxyphenyl)-3-methyl-4-(3,3,3-trifluoropropanesulfonyl)piperazin-2-one
N-methyl-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-N-(pyridin-3-ylmethyl)pyridin-2-amine
N-[2-(benzyloxy)ethyl]-6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[2-methyl-2-(pyrrolidin-1-yl)propyl]amino}methyl)piperidin-2-one
N-(dicyclopropylmethyl)-3-[(4-fluorophenyl)methyl]-1,2-oxazole-5-carboxamide
[(2,2-dimethyloxan-4-yl)methyl](ethyl)[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]amine
5-methyl-3-[(E)-2-phenylethenyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
ethyl 3-[(3-chlorophenyl)methyl]-1-(ethanesulfonyl)piperidine-3-carboxylate
3-(4-methoxy-3,5-dimethylphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine