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3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[1-(4-fluorophenyl)propyl]propanamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
(4aS,7aR)-1-(2-chlorobenzoyl)-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(1-cyclopentylpiperidin-4-yl)methyl][(2,3-dimethoxyphenyl)methyl](oxolan-2-ylmethyl)amine
N-[(2-fluorophenyl)methyl]-3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
5-chloro-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-cyano-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}cyclopropane-1-carboxamide
1-(2,4-difluorophenyl)-3-(ethoxymethyl)-5-(1H-imidazol-1-ylmethyl)-1H-1,2,4-triazole
9-[3-(2-methyl-1H-imidazol-1-yl)butanoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-(thiophen-3-ylmethyl)piperidine
N-{1-[2-oxo-2-(piperidin-1-yl)ethyl]-1H-pyrazol-4-yl}-2-phenoxyacetamide
2,6-dimethoxy-3-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}pyridine
1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(propan-2-yloxy)ethan-1-one
4-ethyl-1-methyl-3-{1-[2-(pyridin-4-yl)ethanesulfonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-1,3-thiazole-4-carboxamide
3-(2-methoxyphenyl)-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)propanamide
N-{1-[7-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}propanamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide
6-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]azetidin-3-yl}pyridine
N'-(4-fluorophenyl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}ethanediamide
N'-cyclopentyl-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]butanediamide
N-(1-benzylpyrrolidin-3-yl)-4-(cyclopentylamino)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-2-(pyrrolidin-3-yl)benzamide
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-(1-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
(5-{1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-imidazol-2-yl}furan-2-yl)methanol
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methylbenzamide
1-cyclopentyl-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-6-oxopiperidine-3-carboxamide
(3S,4R)-4-methyl-1-(5-methylthiophene-2-carbonyl)piperidine-3,4-diol
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
4-(2-methoxyethyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[(2-fluorophenyl)methyl]-1-methyl-6-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}acetamide
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(4-ethoxyphenyl)methyl]piperidine
1-cyclopropyl-N-methyl-5-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidine-3-carboxamide
methyl (2R)-2-[2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamido]propanoate
2-(5-methoxy-1H-indol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
7-(2-hydroxyethyl)-2-[4-(trifluoromethyl)pyrimidin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]oxolane-3-carboxamide
4-(2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}ethyl)morpholine
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
3-(2,5-dimethyl-1H-pyrrol-1-yl)-4,5-dimethyl-N-[(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]thiophene-2-carboxamide
({4-[(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)methoxy]phenyl}methyl)(methyl)(1,2-oxazol-3-ylmethyl)amine
3-(furan-2-yl)-2-{[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]methyl}propan-1-ol
2-methyl-5-{4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
4-(3-methyl-1,2,4-oxadiazol-5-yl)-2-[3-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyridine
5-(5-chloropyrimidin-2-yl)-8-methoxy-2-methylquinoline
N-[(4-methoxyphenyl)methyl]-4-methyl-N-(pyridin-2-ylmethyl)-1H-imidazole-2-carboxamide
2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-4-amine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide