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(1S,4S)-3,3-dimethyl-2-methylidene-N-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)bicyclo[2.2.1]heptane-1-carboxamide
4-(3-chlorobenzoyl)-7-(3,4-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[(3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)carbamoyl}phenyl)amino]acetic acid
(1R,2R,6S,7S)-4-(2,3-difluoro-6-methoxybenzoyl)-4-azatricyclo[5.2.1.02,6]decane
4-(2,2-dimethylpropanoyl)-6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-1,4-diazepan-2-one
2-[(2H-1,3-benzodioxol-4-ylmethyl)(thiophen-2-ylmethyl)amino]butan-1-ol
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(5-chloro-2-methoxybenzoyl)pyrrolidin-3-yl]methanol
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[1-(thiophen-3-yl)propan-2-yl]butanamide
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N3-(4-fluorophenyl)-N5-(oxolan-2-ylmethyl)piperidine-3,5-dicarboxamide
N-[2-(3-methoxyphenyl)-1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]ethyl]-N,3-dimethylbutanamide
N-[3-(5-methyl-4-{[2-(thiophen-2-yl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]-3-(pyridin-3-yl)propanamide
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-amine
3-(4-chlorobenzoyl)-1-[(5-methylfuran-2-yl)methyl]piperidine
2-(1H-imidazol-1-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]ethan-1-one
5-ethyl-5-(3-oxo-3-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}propyl)pyrrolidin-2-one
8-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1-oxa-8-azaspiro[4.5]decane
methyl 4-({[2-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-yl)ethyl]amino}methyl)benzoate
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-4-(pyrrolidin-1-ylmethyl)benzamide
N-cyclopropyl-3-(5-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanamide
1-(oxan-4-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]piperidine-3-carboxamide
8-(2,3-dihydro-1H-inden-2-yl)-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(dicyclopropylmethyl)-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
N-({7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
N,2-dimethyl-N-[2-phenyl-1-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)ethyl]furan-3-carboxamide
2-(2-fluorophenoxymethyl)-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1,3-oxazole-4-carboxamide
1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-3-(1H-pyrazol-4-yl)propan-1-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2-[(2-{[6-(dimethylamino)pyrazin-2-yl]oxy}hex-5-en-1-yl)(methyl)amino]-N,N-dimethylacetamide
5-[1-(2,5-dimethylbenzoyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
6-(1,3-thiazole-5-carbonyl)-N-{[3-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(2S)-1-hydroxy-3-(1H-indol-3-yl)propan-2-yl]propanamide
2-[2-(benzyloxy)phenyl]-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
N-(2-{[2-(4-methoxyphenoxy)ethyl]amino}ethyl)acetamide
methyl({[2-(propan-2-yl)pyrimidin-5-yl]methyl})[1-(1,3-thiazol-2-yl)ethyl]amine
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
2-({[2-(diethylamino)pyridin-3-yl]methyl}amino)pyridine-3-carbonitrile
N-[(2R,3R)-1'-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
5-ethyl-2-(4-phenyl-1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-imidazol-5-yl)pyridine
3-(4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-2,5-dimethylpyrazine
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-methyl-1-[3-(4H-1,2,4-triazol-4-yl)phenyl]urea
3-[(1,4-dimethylpiperazin-2-yl)methyl]-1-[4-(1H-indol-2-yl)phenyl]urea
1-amino-N-[(2-chlorophenyl)methyl]-N-(prop-2-en-1-yl)cyclopropane-1-carboxamide
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propan-1-one
9-[2-(methylsulfanyl)pyrimidin-4-yl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-4-(5-{1-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1H-imidazol-2-yl}thiophen-2-yl)but-3-yn-2-ol
2-ethyl-1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
2-(2,6-dichlorophenyl)-1-[2-(propan-2-yloxy)ethyl]-1H-imidazole
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}pyrrolidin-3-ol