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3-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1'-(2,6-dimethoxypyridine-3-carbonyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine-4-carboxamide
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(2-methoxyphenyl)propanamide
methyl 3-(naphthalene-1-carbonyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[1-({methyl[1-(1,2-oxazol-3-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
1-({1-[6-(4-methylpiperidin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
(2,1,3-benzoxadiazol-4-ylmethyl)(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)methylamine
diethyl({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)amine
5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-propyl-1,2-oxazole-3-carboxamide
2-cyclopentyl-N-(3-{4-[4-(2-methoxyphenoxy)piperidin-1-yl]piperidin-1-yl}phenyl)acetamide
N-[(4-methoxyphenyl)methyl]-N-methyl-5-propyl-1,3,4-oxadiazole-2-carboxamide
(4aS,8aR)-6-(2-methoxyethyl)-1-{[2-(methylsulfanyl)phenyl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
2-{4-[(2,6-difluorophenyl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
4-(3-cyclopentylpropanoyl)-3-(2-hydroxyethyl)piperazin-2-one
2-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-N,N-dimethylaniline
5-[4-(3-chloro-4-fluorophenyl)piperazine-1-carbonyl]-2-(propan-2-yl)pyrimidine
3-{1-[2-(dimethylamino)ethyl]-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl}-N,N-dimethylpiperidine-1-sulfonamide
N-[3-(4-{[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]pyridine-3-carboxamide
4-(1H-imidazol-2-yl)-1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1H-1,2,3-triazole
{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-{[2-(trifluoromethoxy)phenyl]methyl}piperidin-4-ol
(2S,4S)-4-(2,6-difluoro-4-methoxybenzamido)-N-ethyl-1-(2-hydroxyethyl)pyrrolidine-2-carboxamide
N-[1-(4-methylphenyl)ethyl]-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
3-[1-(1H-indole-3-carbonyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
4-methoxy-N-(2-methoxyethyl)-2-{[1-(5-methylhex-5-en-2-yl)piperidin-4-yl]oxy}benzamide
3-({[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amino}methyl)-N-methylpyridin-2-amine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-2-(3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)acetamide
1-(3-chlorophenyl)-4-(6-hydroxyhexyl)piperazin-2-one
1-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]-4-(2H-1,3-benzodioxol-5-ylmethyl)piperazine
N-[2-(morpholin-4-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
2-{4-[(2-fluoro-4-methoxyphenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
(3aS,6aS)-5-cyclohexanecarbonyl-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[1-(6-methylpyridin-2-yl)propan-2-yl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
N-cycloheptyl-2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzamide
4-methoxy-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
5-chloro-N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]furan-2-carboxamide
3-[1-(1,3-benzoxazol-2-yl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
4-chloro-3-[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]-1H-pyrazole
6-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]pyridine-2-carbonitrile
4-chloro-3-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-1,2,3-triazol-4-yl}-1-methyl-1H-indazole
3-{1-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-benzyl-2-methyl-5-(2-methylpropanamido)-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-1,3-benzodiazole-7-carboxamide
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-2-yl)propan-1-one
7-(1,3-benzothiazol-2-yl)-4-(1H-imidazol-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{2-oxo-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
1-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-{2-[1-(pyridin-2-ylmethyl)-1H-1,2,3-triazol-4-yl]phenoxy}ethan-1-ol
5-cyclopropyl-N-(2-{[2-(morpholin-4-yl)ethyl]carbamoyl}phenyl)-1,2-oxazole-4-carboxamide