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N'-cyclopentyl-N-methyl-N-(1H-pyrazol-5-ylmethyl)butanediamide
1-methyl-3-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazol-5-one
1-{3-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-[methyl(piperidin-4-yl)amino]ethan-1-one
2-methyl-4-(2-methylphenyl)-1-[4-(piperidine-1-carbonyl)pyridin-2-yl]piperazine
3-(2-methylphenoxymethyl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-3-ol
2-amino-4-(1-benzofuran-2-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
2-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxo-N-phenylacetamide
(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-amino-2-{4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}pyrimidine-5-carbonitrile
2-amino-3-ethyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-(azepan-1-yl)-3-(2-methoxy-4-{[(3-phenylpropyl)amino]methyl}phenoxy)propan-2-ol
N-(2-methoxyethyl)-1-(methoxymethyl)-N-(pyridin-4-ylmethyl)cyclobutane-1-carboxamide
1-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}urea
1-cyclohexyl-N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]piperidine-4-carboxamide
methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}amine
5-ethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
3-(azepane-1-carbonyl)-N-methyl-N-(oxolan-3-ylmethyl)benzene-1-sulfonamide
1-ethoxy-3-{[5-(naphthalen-2-yl)-1,2,4-triazin-3-yl]amino}propan-2-ol
4-[2-(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-2-yl)ethyl]phenol
6-chloro-2-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]quinoline
4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-2-(morpholin-4-ylmethyl)-1,4-oxazepane
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
1-(3-phenyl-1H-pyrazole-4-carbonyl)-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
8-fluoroquinoline-2-carboxamide
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
5-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyrazin-2-ol
6-(6-fluoroquinolin-8-yl)pyridine-3-carboxylic acid
{2,2-dimethyl-3-[4-(4-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propyl}dimethylamine
N4-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-6-methyl-5-(prop-2-en-1-yl)pyrimidine-2,4-diamine
6-[({[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}amino)methyl]-1,4-oxazepan-6-ol
N-(3-methoxypropyl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
5-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]quinoline
5-chloro-7-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1-benzofuran-2-carboxylic acid
1-[3-(2-phenylethyl)piperidin-1-yl]pent-4-en-1-one
1-(1,2,3,4-tetrahydronaphthalen-1-yl)-3-(1,2,3-thiadiazol-5-yl)urea
1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-4-(1H-imidazol-2-yl)piperidine
4-[2-({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}amino)ethyl]phenol
1-(2-{1-[1-(4-methylphenyl)cyclopropanecarbonyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
N-cyclobutyl-6-(2,5-dimethylfuran-3-yl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(1R,5R)-6-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-amino-4-[2-(benzylamino)pyrimidin-5-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-butyl-11-[methyl(2-methylpropyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-1-phenylcyclohexane-1-carboxamide
N-(propan-2-yl)-6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-4-amine
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}urea
(3aR,5R,6S,7aS)-2-(6-methyl-2-phenylpyrimidin-4-yl)-octahydro-1H-isoindole-5,6-diol
5-methyl-1-{2-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
N-(3,4-dimethylphenyl)piperidin-3-amine