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2-{5-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-3-(1H-imidazol-1-ylmethyl)piperidine
2-[(2S)-2-aminobutanoyl]-N-(5-methyl-1,2-oxazol-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-{1-[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}ethan-1-one
N-cyclopropyl-2-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}pyridine-4-carboxamide
methyl 2-(1-{1-[2-(4-chlorophenyl)ethyl]-6-oxopiperidin-3-yl}-N-methylformamido)acetate
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-methylthiophene-2-carboxamide
2-(9-{[2-(ethylamino)pyrimidin-5-yl]methyl}-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl)acetic acid
4-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
(3R,4R)-1-{[3-(benzyloxy)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
2-{4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
7-(pyridin-3-yl)-4-[4-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-methoxy-3-methyl-2-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1H-indole
2-[5-(2,1,3-benzoxadiazol-4-yl)-4-phenyl-1H-imidazol-1-yl]acetic acid
N-ethyl-5-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
4-{2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
3-(tert-butylsulfamoyl)-5-{[(2E)-4-methylpent-2-en-1-yl]amino}-N-[(1-methylpiperidin-3-yl)methyl]benzamide
1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-2-(pyrrolidin-1-yl)ethan-1-one
1-(2,6-difluorobenzenesulfonyl)-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
3-{[2-(5-chlorothiophen-2-yl)-1H-imidazol-1-yl]methyl}-4-propyl-4H-1,2,4-triazole
1-[(3-methoxyphenyl)methyl]-N-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-amine
[(4-{[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]urea
1-[(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)methyl]-3,5-dimethyl-1H-pyrazole
7-[(3,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
({4-[3-(2-methoxyethyl)-1-[(2-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl]-1,3-thiazol-2-yl}methyl)dimethylamine
3-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]phenol
1-{1-[5-(3-chlorophenyl)-1,2,4-triazin-3-yl]piperidin-3-yl}-3-methylbutan-1-one
3-[(cyclopentylamino)methyl]-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
N-[3-(3-chlorophenoxy)propyl]-N-methyl-2-(pyrrolidin-3-yl)acetamide
1-ethyl-4-{[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-3-methyl-1H-pyrazole
4-(2-methyl-2-{1-[(5-methylpyrazin-2-yl)methyl]-1H-imidazol-2-yl}propyl)morpholine
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-[(1-ethylpiperidin-4-yl)amino]-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
4-(1H-imidazol-2-yl)-1-[2-(1H-pyrrol-1-yl)benzoyl]piperidine
10-methoxy-5-[3-(1H-pyrazol-1-yl)benzoyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
{3-[(3-chlorophenyl)methyl]-1-[(3,5-dimethoxyphenyl)methyl]piperidin-3-yl}methanol
3-(2-methylpropyl)-5-(2,3,4-trimethoxyphenyl)-1H-1,2,4-triazole
1-(cyclohexylmethyl)-3-{[(2,3-dihydroxypropyl)amino]methyl}-6,7-dimethoxy-1,2-dihydroquinolin-2-one
3-(3-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]propan-1-one
N-cyclohexyl-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2S,4R)-4-amino-N-methyl-1-(9-oxo-9,10-dihydroacridine-4-carbonyl)pyrrolidine-2-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-3-carboxamide
{1-[(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
1-ethyl-N-(3-methylbutyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(3-methylbutyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-[(3-hydroxypiperidin-1-yl)methyl]-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
1-{2-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propan-1-one
N-({1-[3-(furan-2-yl)propanoyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
2-{[(3R,5S)-1-{[4-(benzyloxy)phenyl]methyl}-5-(4-methyl-1,4-diazepane-1-carbonyl)pyrrolidin-3-yl]sulfanyl}-1H-1,3-benzodiazole