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2-[(2,6-dichlorophenyl)methyl]-5-(2-ethylpyrrolidine-1-carbonyl)pyrimidin-4-ol
5-{1-[(4-fluorophenyl)methanesulfonyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
2-[(1S,5R)-3-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
1-(pyridin-3-yl)-4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazine
N-[2-(1-methylpiperidin-3-yl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-amine
2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}acetamide
N5-(2,3-dihydro-1H-inden-1-yl)-N6-(2-methoxyethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-[2-(methylsulfanyl)benzoyl]-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidine
N-[(5-chlorothiophen-2-yl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2,2-diphenyl-1-[4-(1,3-thiazol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]ethan-1-ol
3-{[methyl(prop-2-en-1-yl)amino]methyl}-N-(1-propyl-1H-1,2,4-triazol-3-yl)benzamide
2-[1-(cyclopropylmethyl)-4-(6-methyl-2-propylpyrimidin-4-yl)piperazin-2-yl]ethan-1-ol
2-[(1S,5R)-6-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-(2-methoxyphenyl)-N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)propanamide
N-cycloheptyl-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
8-[2-(3,4-dimethoxyphenyl)acetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[1-(3-ethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-2-methyl-6-(pyrrolidin-1-yl)pyrimidine
1-butyl-4-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}piperazin-2-one
3-oxo-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
(3S)-N,N-dimethyl-1-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]azepan-3-amine
N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-1-methyl-1H-indole-6-carboxamide
4-[(2,3-dimethyl-1H-indol-7-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)oxane-2-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-4-methyl-1H-imidazole-5-carboxamide
2-{4-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
3-(1,3-benzothiazol-2-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}propanamide
2-ethoxy-1-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
1-(2-methoxyethyl)-4-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperazine
N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-3-(3-phenoxypropanoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-methyl-N-(oxan-2-ylmethyl)propanamide
N-[2-(2-chloro-6-fluorophenyl)ethyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
5-ethyl-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)-1,3-oxazole-4-carboxamide
4-methoxy-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidine
N-[2-(1H-1,3-benzodiazole-1-carbonyl)phenyl]pyridine-2-carboxamide
2-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
1-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(2-methoxyphenyl)propan-1-one
N-(4-{4-[(cyclopentylformamido)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)-5-(methoxymethyl)furan-2-carboxamide
7-fluoro-N-[1-(1H-imidazol-1-yl)butan-2-yl]-2-methylquinoline-4-carboxamide
N-[2-(6-methylpyridin-2-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
ethyl 3-benzyl-1-(4-methoxybenzenesulfonyl)piperidine-3-carboxylate
1-butyl-3-methyl-4-(piperidin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
ethyl 1-benzyl-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-{2-[(pyridin-4-ylmethyl)amino]pyrimidin-4-yl}pyrrolidin-3-ol
2-methyl-8-[(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)sulfonyl]-2,8-diazaspiro[4.5]decan-3-one