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1-(6-methyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-benzamido-1-cyclopentyl-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
8-(1-methyl-1H-pyrrole-2-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-(9H-fluoren-9-yl)propanamide
6-[(diethylamino)methyl]-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(2-hydroxyethyl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1H-1,3-benzodiazole-5-carboxamide
4-(cyclohexylmethyl)-3-(1-methylpiperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(1-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}piperidin-3-yl)methanol
1-(2-ethoxyethyl)-N,3-dimethyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-pyrazole-5-carboxamide
5-(methoxymethyl)-N-{3-methyl-1-[7-(pyridin-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}furan-2-carboxamide
3-[(5-chlorothiophen-2-yl)methyl]-8-methyl-3,4-dihydroquinazolin-4-one
1-[2-chloro-5-(morpholine-4-carbonyl)phenyl]-3-{2-[(2R)-pyrrolidin-2-yl]ethyl}urea
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
1-[2-(3,4-dimethoxyphenyl)ethyl]-5-[2-(ethylamino)ethyl]pyrrolidin-2-one
3-{[(1,4-dithiepan-6-yl)amino]methyl}-6-ethyl-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(1S,5R)-3-(2-methoxypyridine-4-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl}-1H-1,3-benzodiazole
N-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
ethyl 1-[(2S)-5-oxopyrrolidine-2-carbonyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
(3S,4S)-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
1-[cyclohexyl(methyl)amino]-3-[2-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
(4aR,7aS)-1-acetyl-4-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{[4-(2-{1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-2-yl}ethoxy)phenyl]methyl}piperazine-1-carbaldehyde
N-(4-{1-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-1H-1,2,3-triazol-4-yl}phenyl)acetamide
(4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}morpholin-2-yl)methanamine
2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[2-(6-methylpyridin-2-yl)ethyl]acetamide
(3R,4R)-4-(hydroxymethyl)-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-3-ol
2-(4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-1-(2-methylpropyl)piperazin-2-yl)ethan-1-ol
(1S,5R)-6-(3-ethyl-1,2-oxazole-5-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
(3S,4S)-1-(4-methylpyrimidin-2-yl)-4-(piperidin-1-yl)pyrrolidin-3-ol
4-amino-N-[3-(phenylsulfanyl)propyl]pyridine-2-carboxamide
2-[(1S,5R)-3-(3-fluoropyridine-4-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
4-[7-(3-hydroxypyridine-2-carbonyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
6-methyl-4-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-1-[2-(methylsulfanyl)phenyl]piperazin-2-one
N-[5-(4-methylpiperazine-1-carbonyl)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]thiophene-2-carboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-yl]cyclopropanecarboxamide
2-[4-(3-methylphenyl)piperazin-1-yl]-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
N,6-dimethyl-N-[(1-methylpyrrolidin-3-yl)methyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(3,5-dimethoxyphenyl)methyl]piperidine
N5-benzyl-N6-(pyridin-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-(2-phenylethyl)-4-(thiophen-3-ylmethyl)morpholine
5-methyl-2-(4-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}piperidin-4-yl)pyridine
1-{2-hydroxy-3-[2-methoxy-4-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
4-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1λ6-thiane-1,1-dione
N-[1-(4-fluorophenyl)-2-hydroxyethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
4-methyl-N-(2-methyl-1,3-benzothiazol-5-yl)-1,2,3,6-tetrahydropyridine-1-carboxamide
N-[3-(5-methyl-4-{[(5-methyl-3-phenyl-1,2-oxazol-4-yl)formamido]methyl}-1,3-oxazol-2-yl)phenyl]pyridine-4-carboxamide
2,6-dimethyl-N-[1-(4-methylphenyl)-5-oxopyrrolidin-3-yl]quinoline-4-carboxamide