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4-[3-(benzyloxy)propyl]-1,3λ6,4-oxathiazinane-3,3-dione
5-(2,6,8-trimethylquinoline-4-carbonyl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
3-benzoyl-1-[1-(methylsulfanyl)propan-2-yl]piperidine
4-(4-fluorophenyl)-1-{1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carbonyl}-1,2,3,6-tetrahydropyridine
1-{1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]piperidin-3-yl}pyrrolidin-2-one
2-[2-(2,3-dimethylphenoxy)ethyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(benzyloxy)-1-[(2R)-oxolane-2-carbonyl]piperidine
2-(3-chlorophenyl)-N-[4-(4-{methyl[2-(oxan-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
2,2-dimethyl-6-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-3,4-dihydro-2H-pyran-4-one
4-chloro-3-({[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]carbamoyl}amino)-N-methylbenzamide
5-(2-benzyl-1,3-thiazol-4-yl)-3-ethyl-1,2,4-oxadiazole
1-cyclopropanecarbonyl-4-[4-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-6-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
(4-{[1-(2-methoxy-5-methylbenzenesulfonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
(1R,9aR)-1-(3,4,5-trimethoxyphenoxymethyl)-octahydro-1H-quinolizine
[2-(1H-imidazol-1-yl)ethyl]({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})methylamine
2,6,8-trimethyl-N-[3-(3-oxopiperazin-1-yl)propyl]quinoline-4-carboxamide
4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrimidin-2-amine
3-(2H-1,3-benzodioxol-5-yl)-5-(furan-3-ylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-N,6-dimethyl-4-oxo-N-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-(1,3-thiazol-5-ylmethyl)-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
4-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}-1-(1,3-thiazole-5-carbonyl)piperidine
1-(3-cyano-4-methoxyphenyl)-3-[1-(thian-4-yl)piperidin-4-yl]urea
(3aR,6aR)-2-(2-aminopyrimidin-4-yl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)[(3-methylphenyl)methyl]amine
4-(3-chloropyridin-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-3-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}urea
7-[(2-chloro-4-hydroxyphenyl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-[2-(1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
4-{5-[(3-fluoro-2,4-dimethylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-(prop-2-en-1-yl)-1H-pyrazole
N-[2-(pyridin-3-yloxy)ethyl]-1-benzothiophene-5-carboxamide
2-amino-4-phenyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidine-5-carboxamide
(2S,4R)-4-(3-chlorothiophene-2-amido)-N-ethyl-1-(3-methylbut-2-en-1-yl)pyrrolidine-2-carboxamide
N-methyl-5-{[3-(3-phenylpropanoyl)piperidin-1-yl]methyl}furan-2-carboxamide
2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-7-methyl-4H-chromen-4-one
4-ethyl-5-methyl-2-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}pyrimidine
2-(dimethylamino)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-2,3-dihydro-1H-indene-2-carboxamide
4-{1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidin-4-yl}-6-(pyrrolidin-1-yl)pyrimidine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-1-(propan-2-yl)piperidine-4-carboxamide
6-ethyl-N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2-methylquinoline-4-carboxamide
N-[2-(azepan-1-yl)ethyl]-N-ethyl-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propanamide
1-benzyl-4-{[4-(4-methylpiperidine-1-carbonyl)-1,3-oxazol-2-yl]methyl}piperazine
2-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}acetamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1-methyl-1H-1,3-benzodiazole-5-carboxamide
1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-4-(thiophene-2-carbonyl)-1,4-diazepan-2-one
1-cyclopentyl-N-methyl-6-oxo-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidine-3-carboxamide
N-({7-[(2-chloro-3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide