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3-(1,2-oxazinan-2-yl)-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]propanamide
1-cyclohexyl-4-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-{3-[3-(4-chloro-2-methylbenzoyl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
[(6-chloroquinolin-2-yl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
3-(2-fluorophenyl)-5-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(2-oxopyrrolidin-1-yl)propanamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
2-(2,5-difluorophenyl)-2-{2-[1-(propan-2-yl)piperidin-4-yl]acetamido}acetic acid
N,N,2-trimethyl-4-[4-(prop-2-en-1-yl)piperazin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-3-(pyridin-3-yl)-N-(pyridin-3-ylmethyl)propanamide
2-[2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
6-fluoro-4-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
N-ethyl-15-methyl-13-oxo-9-(pyridin-3-yl)-4-(trifluoromethyl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
(4aR,8aS)-1-[5-(methoxymethyl)furan-2-carbonyl]-6-[4-(trifluoromethyl)benzoyl]-decahydro-1,6-naphthyridine
N-[(1-ethylpyrrolidin-2-yl)methyl]-5-(1H-indole-5-carbonyl)-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-methyl-2-{1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
N-({1-[(3,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)-1H-1,2,4-triazole-5-carboxamide
4-({4-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]furan-2-yl}methyl)morpholine
methyl (2S,4S,5R)-4-(4-ethylpiperazine-1-carbonyl)-1,2-dimethyl-5-(2-methylphenyl)pyrrolidine-2-carboxylate
1-(cyclohex-3-en-1-ylmethyl)-4-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one
2-(3-methylbutyl)-8-(pyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
7-(5-chloropyridin-2-yl)-4-[(3-hydroxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(3-methoxyphenyl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)-1H-pyrazole-4-carboxamide
4-hydroxy-N-propyl-2-(pyridin-2-yl)-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
4-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}morpholine
(4aS,8aR)-6-(5-chloropyridin-2-yl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
(3aS,6aS)-5-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[1-(4-methoxyphenyl)ethyl]methylamine
(1S,5R)-3-(pyridin-2-ylmethyl)-6-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N,N-diethyl-3-[({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amino)methyl]pyridin-2-amine
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-[4-(methylsulfanyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
3-{[5-(1-acetylpiperidin-2-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}benzonitrile
2-[3,5-bis(trifluoromethyl)phenyl]-N-ethyl-4-hydroxy-N-methylpyrimidine-5-carboxamide
3-{[2-(4-methoxyphenoxy)ethyl]amino}-2,2-dimethylpropan-1-ol
1'-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]spiro[indene-1,4'-piperidine]
(2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-1,3-thiazol-4-yl)methanol
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
3-{methyl[1-(1,2-oxazol-3-yl)ethyl]sulfamoyl}-N-(prop-2-en-1-yl)benzamide
2-(dimethylamino)-7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
8-[(4-methyl-1,3-thiazol-5-yl)methyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[4-(1-benzothiophen-5-ylmethyl)-1-methylpiperazin-2-yl]ethan-1-ol
2-(2H-1,3-benzodioxol-5-yl)-3-methoxypyrazine
(3S)-3-benzyl-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-2-one
1-methyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(3-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]piperidine-4-carbonitrile
3-(3-fluoro-2-methylphenyl)-1-[(3-methoxyphenyl)methyl]-1-(3-methoxypropyl)urea
1-[(2-methoxyphenyl)methyl]-4-[5-(pyridin-3-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
2-butyl-8-(3-hydroxy-2-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one