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3-({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)amino)propan-1-ol
N-[(1-cyclopentylpiperidin-3-yl)methyl]-3-methoxy-N-[2-(piperidin-1-yl)ethyl]propanamide
(2S)-1-[4-(4-chlorophenyl)butanoyl]pyrrolidine-2-carboxylic acid
N-[3-(azepan-1-yl)-2-hydroxypropyl]-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
3-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,5R)-N-[2-(1H-imidazol-4-yl)ethyl]-1-(2-phenylethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-ethyl-2,2-dimethyloxan-4-amine
4-(2-fluorophenoxy)-1-(4-methyl-1H-imidazole-2-carbonyl)piperidine-4-carboxylic acid
3-(2-cyclopropylacetyl)-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
ethyl 1-cyclobutyl-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
8-[3-(propan-2-yl)-5-(1H-1,2,4-triazol-5-yl)-1H-1,2,4-triazol-1-yl]quinoline
4-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}phenol
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,1-dimethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-(3-cyano-4,5-dimethylthiophen-2-yl)-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
7-[(2,3-difluorophenyl)methyl]-2-(3,4-dimethylbenzoyl)-2,7-diazaspiro[4.5]decane
N-(furan-2-ylmethyl)-3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxamide
1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-3-yl)propan-1-one
N-(2-methoxyethyl)-1-[1-(quinolin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
1-(2-phenylethyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propanamide
5-[bis(prop-2-en-1-yl)amino]-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-amine
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-1-[4-(quinazolin-2-yl)piperazin-1-yl]ethan-1-one
6-methyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}pyridine-2-carboxamide
(3R,4S)-1-[1-(2-fluorophenyl)piperidin-4-yl]-3,4-dimethylpiperidin-4-ol
N-[(2S,4R,6S)-2-ethyl-6-(3-phenoxyphenyl)oxan-4-yl]acetamide
2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-cyclopropylacetamide
8-(5-methoxy-1H-indole-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-cyclopropyl-3-({[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}sulfamoyl)benzamide
N-({7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
N-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
methyl 2-(1-{3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanoyl}-3-oxopiperazin-2-yl)acetate
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-[4-(2-methylphenoxy)piperidin-1-yl]ethan-1-one
3-methyl-1-(2-oxo-2-{4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}ethyl)pyrrolidin-2-one
2-methanesulfonyl-N-[2-(3-phenylpropoxy)phenyl]acetamide
N-cyclopropyl-1-[1-(1H-indol-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-(5-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propyl}-1,2,4-oxadiazol-3-yl)pyridine
1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}-4-(propan-2-yl)piperazine
1-(3-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
(3S,4R)-1-(1H-imidazol-2-ylmethyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
(1-{[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)methanol
1-[3-(oxan-4-yl)-1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-6-azaspiro[2.5]octane
1-(carbamoylmethyl)-N-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]methyl}piperidine-3-carboxamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pent-4-enamide
4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methylpyrimidine
N-[2-(furan-2-yl)ethyl]-7-(3-methoxypropanamido)-1-methyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
4-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2,2-diphenylbutanenitrile
4-{5-[4-(3-methylphenoxy)piperidine-1-carbonyl]pyrimidin-2-yl}morpholine
1-(4-methyl-1,3-thiazol-2-yl)-3-(2-methylphenyl)piperidine