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4-(1-benzoxepine-4-carbonyl)-2-(trifluoromethyl)morpholine
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carboxamide
5-(2-methylphenoxymethyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
({4-ethyl-5-[1-(3-fluoro-4-methoxybenzoyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
9-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2,6-dimethoxy-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]pyridine-3-carboxamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[3-(pyridin-3-yl)propyl]pyrrolidine-3-carboxylic acid
1-[1,5-bis(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
4-(9H-fluoren-2-ylmethyl)piperazine-2-carboxylic acid
8-methoxy-3-{[1-(2-phenylethyl)piperidin-3-yl]methyl}-3,4-dihydroquinazolin-4-one
2,2-dimethyl-N-(1-{1-[2-(2-methylphenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
9-[4-(hydroxymethyl)benzoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-4-[(3-fluorophenyl)methyl]piperazin-2-one
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[2-(pyrrolidine-1-sulfonyl)ethyl]acetamide
N-cyclopropyl-3-[5-(2,6-dimethylpyrimidine-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropylnaphthalene-1-carboxamide
2-[1-(cyclohexylmethyl)-4-[(2,4,6-trimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-(1-{[1-(2-ethoxyethyl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}-1H-pyrazol-5-yl)acetamide
2-[(1-ethylpyrrolidin-2-yl)methyl]-4-(1,4-oxazepane-4-carbonyl)-2,3-dihydro-1H-isoindol-1-one
ethyl 4-[6-(quinolin-7-ylmethyl)-6-azaspiro[2.5]octane-1-carbonyl]piperazine-1-carboxylate
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-(6-hydroxy-1,4-oxazepan-4-yl)ethan-1-one
(4aR,7aS)-1-[(3-hydroxyphenyl)methyl]-4-(2-phenylethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[5-(5-phenylpentanoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
4-[2-(1-ethyl-1H-1,2,4-triazol-5-yl)-1H-imidazol-1-yl]-N,N-dimethylaniline
1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[3-(trifluoromethyl)phenyl]piperazine
3-{1-[5-(4-methylphenyl)-1H-pyrazole-3-carbonyl]piperidin-2-yl}pyridine
1-(dimethylsulfamoyl)-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
2-[(4aR,7aS)-6,6-dioxo-4-(2-propoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
(3S,4R)-1-(2,6-dimethoxybenzoyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
5-[3-(1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazol-3-yl)phenyl]pyrimidine
5-(morpholin-4-yl)-2-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,3-dihydropyridazin-3-one
N-[3-(1H-imidazol-1-yl)propyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
5-(2-{[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethyl)-1,3,4-thiadiazol-2-amine
1-(4,7-dimethylquinazolin-2-yl)-N-(oxan-4-yl)azepan-4-amine
N,N-diethyl-4-({[2-(1H-imidazol-4-yl)ethyl]carbamoyl}amino)-3-methylbenzamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-4-(1H-pyrazol-1-yl)butanamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
5-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
5-[4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]quinoxaline
[(3R,4S)-1-[(5-fluoro-2-methoxyphenyl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]furan-2-carboxamide
(2R)-N-(4-chloro-2-methoxy-5-methylphenyl)-2-(hydroxymethyl)pyrrolidine-1-carboxamide
(1S,5R)-6-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-2-{4-[6-(trifluoromethyl)pyridin-2-yl]-1H-pyrazol-1-yl}acetamide
4-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}-3-(3,4,5-trimethoxyphenyl)-1H-pyrazole
1-benzyl-4-(1H-pyrrole-2-carbonyl)-1,4-diazepan-6-ol
4-(5-tert-butyl-2-methoxybenzenesulfonyl)piperazine-2-carboxylic acid
6-fluoro-2-{[2-(2-methoxyethyl)morpholin-4-yl]methyl}quinolin-4-ol