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2-{[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}-1-(pyridin-3-yl)ethan-1-ol
(2R)-N-{2-[(pyridin-3-yl)amino]ethyl}oxolane-2-carboxamide
1-[2-(cyclohex-1-en-1-yl)ethyl]-2-(oxolan-3-yl)-1H-imidazole
2-(dimethylamino)-2-(2-fluorophenyl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide
N5-tert-butyl-N3-methyl-4-oxo-1-(propan-2-yl)-N3-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
3-methoxy-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine
4-(piperidin-1-ylmethyl)-N-[2-(1,3-thiazol-2-yl)ethyl]benzamide
N-[3-(5-cyano-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carbonyl)phenyl]butanamide
(3aS,6aR)-3-cyclopentyl-5-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}oxolane-3-carboxamide
benzyl(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)(1,3-thiazol-2-ylmethyl)amine
N-[1-(3-phenylpropyl)piperidin-3-yl]-2-(pyridin-2-ylsulfanyl)acetamide
N-[2-(4-fluorophenyl)ethyl]-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2-(thiophen-3-yl)acetamide
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(propan-2-yloxy)propan-1-one
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
N-(pyridin-3-ylmethyl)-3-[1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-4-yl]propanamide
2-{[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]methyl}benzonitrile
(1S,5R)-3-[2-(methylamino)pyridine-4-carbonyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(2,4-difluorophenoxymethyl)-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,2-oxazole-3-carboxamide
1-(naphthalen-2-yl)-4-(1H-pyrrole-2-carbonyl)piperazine
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
3-ethoxy-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]propanamide
4-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}-1-(2-methylpropyl)piperidine
1-(4,7-dimethylquinazolin-2-yl)-N-[1-(thiophen-2-yl)propan-2-yl]piperidine-4-carboxamide
1-ethyl-4-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-2,3-dihydro-1H-inden-2-yl}piperazine
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[2-(furan-2-ylmethoxy)phenyl]-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
1-tert-butyl-4-[4-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]pyrrolidin-2-one
2-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-phenyl-1,2-dihydrophthalazin-1-one
4-methyl-6-{4-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperazin-1-yl}pyrimidin-2-amine
N,N-dimethyl-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
4-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}-2-(trifluoromethyl)pyrimidine
methyl 6-({[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]carbamoyl}amino)-1,2,3,4-tetrahydroquinoline-1-carboxylate
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-3-(trifluoromethyl)benzene-1-sulfonamide
(4aR,8aS)-6-(adamantan-2-yl)-1-(2H-1,3-benzodioxol-5-ylmethyl)-decahydro-1,6-naphthyridin-2-one
[5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-2-fluorophenyl]methanol
2-(dimethylamino)-2-(2-methylphenyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]acetamide
N-(1-benzylpiperidin-4-yl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
5-[methyl(2-phenylethyl)amino]-2-[3-(morpholin-4-yl)propyl]-2,3-dihydropyridazin-3-one
(3S,4R)-4-(2-methoxyphenyl)-1-(oxane-4-carbonyl)pyrrolidine-3-carboxylic acid
1-{2-[1-(4-methylpyridine-3-carbonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
4-(2-ethyl-6-methylpyrimidin-4-yl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-methyl-9-oxo-N-(thiophen-3-ylmethyl)-9,10-dihydroacridine-4-carboxamide
5-(2-butyl-1H-imidazol-4-yl)-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-phenyl-1H-imidazole
methyl(pyrazin-2-ylmethyl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
N-(4-methoxy-2-methylphenyl)-3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,5,7-trimethylpyrido[2,3-d]pyrimidin-4-amine
N-[(4-hydroxy-1-{[2-(methylsulfanyl)phenyl]methyl}azepan-4-yl)methyl]pyrrolidine-1-carboxamide
3-(1H-imidazol-1-yl)-1-[4-(2-methoxyphenoxy)piperidin-1-yl]butan-1-one
4-[3-(3-chlorophenyl)-3-phenylpropanoyl]piperazin-2-one