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ethyl 4-(3-phenylpropyl)-1-(pyridin-3-ylmethyl)piperidine-4-carboxylate
1-(2-cyclohexylethyl)-3-hydroxy-3-[(4-phenylpiperazin-1-yl)methyl]piperidin-2-one
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
3-[2-(morpholin-4-yl)-2-oxoethyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-one
(1R,2R)-N-methyl-2-phenyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}cyclopropane-1-carboxamide
2-[6-(cyclopentylamino)pyridazin-3-yl]benzamide
1-(2-{methyl[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amino}ethyl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-(azepane-1-sulfonyl)-5-(pyridin-3-yl)benzoic acid
1-methyl-1-(thiophen-3-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)urea
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(pent-2-yn-1-yl)piperidine
3-[(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]phenol
N-benzyl-5-{imidazo[1,2-a]pyridine-2-carbonyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2R,3S,6R)-5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
2-methyl-8-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-[1-(2-phenoxyacetyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
methyl({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)(thiophen-2-ylmethyl)amine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidine
4-(4-methoxyphenyl)-2-methyl-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperazine
[4-({5-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-4-phenyl-1H-imidazol-1-yl}methyl)oxan-4-yl]methanol
2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrazine
ethyl 1-(2H-1,3-benzodioxole-5-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
2-(2,4-dichlorophenoxy)-N-(isoquinolin-5-ylmethyl)-N-methylacetamide
2-[(tert-butylsulfanyl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{[5-(2-fluorobenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}azocane
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(2,2-dimethyloxan-4-yl)-6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(1-methyl-1H-pyrazol-4-yl)-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
5-(2,6-difluorophenoxymethyl)-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
5-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]pyrimidine-2,4-diol
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)acetamide
2-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenol
1-cyclopropyl-5-{4-[3-(trifluoromethyl)phenoxy]piperidine-1-carbonyl}piperidin-2-one
2-(4-hydroxyphenyl)-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
1-(2-cyclohexylethyl)-3-hydroxy-3-({[2-(1H-1,2,3-triazol-1-yl)ethyl]amino}methyl)piperidin-2-one
N-[(2-ethoxyphenyl)methyl]-4-methyl-5-(1-methyl-1H-pyrazol-3-yl)-1,3-thiazol-2-amine
5-(1H-imidazol-2-yl)-2-(2-methylphenyl)pyrimidine
(2-{2-[1-(4-fluoro-3-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-(2-methylpropyl)-1-[(1s,4s)-4-{[(3-ethoxy-2-hydroxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
8-[2-(2,3-dimethylphenoxy)ethyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
2-ethoxy-5-(2-{[(4-methylpyridin-2-yl)methyl]amino}pyrimidin-4-yl)benzoic acid
1-(oxan-4-yl)-4-[3-(oxolan-3-yl)-1-propyl-1H-1,2,4-triazol-5-yl]piperidine
4-{[2-(1H-indol-3-yl)ethyl]amino}-N-(1-methoxybutan-2-yl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-({[(2-butoxy-3-methoxyphenyl)methyl]amino}methyl)-3,5-dimethylpyridin-4-ol
2-{2-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}quinoxalin-2-amine
1-[1-(2-hydroxypyridine-3-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
2-[(3,4-dimethoxyphenyl)methyl]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1,3-benzoxazole-6-carboxamide
2-chloro-N-ethyl-4,5-difluoro-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]benzamide