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methyl({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl})(1,3-thiazol-4-ylmethyl)amine
methyl 3-[(cyclobutylformamido)methyl]-5-[2-(thiophen-3-yl)acetamido]benzoate
8-cyclopentyl-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
5-(methoxymethyl)-N-({7-[(4-phenyl-1,3-thiazol-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)furan-2-carboxamide
1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
3-methyl-5-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-2-yl)-1H-1,2,4-triazole
methyl 1-benzyl-3-cyclopropaneamido-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1S,5R)-3-benzoyl-6-(naphthalene-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{1-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]piperidin-4-yl}piperidin-3-ol
2-{5-[(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)methyl]-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl}acetic acid
4-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
4-[(2S)-1-acetylpyrrolidine-2-carbonyl]-6-(benzyloxy)-1-cyclohexyl-1,4-diazepan-2-one
6-(3-methoxypyrrolidin-1-yl)-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-amine
N-(1-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
8-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-benzyl-N-(3-hydroxy-2-methylpropyl)-2-[(2-oxo-2H-chromen-7-yl)oxy]acetamide
5-(1-benzofuran-2-yl)-N-methyl-N-[2-(4-methylphenoxy)ethyl]-1,2,4-triazin-3-amine
4-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N-methyl-5-(1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-methyl-N-phenyl-2-[(1R,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
2-[({1-azabicyclo[2.2.2]octan-3-yl}amino)methyl]-4-(pyridin-2-yl)phenol
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-3-yl}propanamide
2,6-dimethyl-5-(2-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-3-(2-oxoimidazolidin-1-yl)benzamide
(3aS,6aS)-2-cyclohexyl-5-{[4-(methylcarbamoyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-3-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]urea
2-(1-butyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
6-[2-(methylsulfanyl)benzoyl]-N-[3-(2-oxoimidazolidin-1-yl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
2-[(2-{methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]carbamoyl}phenyl)amino]acetic acid
N-[(4-fluorophenyl)methyl]-3-(1,2-oxazolidin-2-yl)-N-(oxolan-2-ylmethyl)propanamide
1-{4-[(2-fluoro-5-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2-phenylethan-1-ol
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-(piperidin-1-yl)ethan-1-one
(3S,4R)-1-(5-fluoro-3-methyl-1H-indole-2-carbonyl)-4-methyl-3-(2-methylpropyl)piperidin-4-ol
8-chloro-2-[({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)methyl]quinolin-4-ol
propan-2-yl (4aS,7aR)-6,6-dioxo-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
1-[(2-methoxyphenyl)methyl]-4-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]piperazine
2-[(cyclopropylmethyl)sulfanyl]-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
N-[1-({[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
4-ethyl-3-{1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1-{1-[3-(1H-indol-3-yl)propanoyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperidine-3-carboxamide
2-cyclobutyl-1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]ethan-1-one
N-[3-(4-fluorophenyl)propyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
1-(3,3-diphenylpiperidin-1-yl)-2-(morpholin-3-yl)ethan-1-one
1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
3-(2-phenylethyl)-7-(2-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N,1,3-trimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[(3-methoxyphenyl)methyl]-2-(4-methylpiperazin-1-yl)-N-(prop-2-en-1-yl)propanamide