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8-(2-hydroxypropyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-(cyclopropylmethyl)-4-{imidazo[1,2-a]pyridine-3-carbonyl}-2-(propan-2-yl)-1,4-diazepane
1-[1-(1H-pyrrole-3-carbonyl)piperidin-4-yl]piperidin-3-ol
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
2-{3-[1-(2-fluoro-4-methylphenyl)-1H-imidazol-2-yl]phenoxy}acetamide
(2S)-N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-acetamido-4-(methylsulfanyl)butanamide
9-methoxy-4-[(3-methylphenyl)methyl]-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-cyclopentyl-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(1R,9S)-5-amino-3-[2-(furan-2-yl)pyrimidin-5-yl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
1-({1-[2-(1H-imidazol-5-yl)ethyl]-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl}methyl)-1,2-dihydropyridin-2-one
3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
4-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-chlorophenol
[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl](methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
(2R,6R)-4-(trimethyl-1H-pyrazole-4-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-1λ6-thiomorpholine-1,1-dione
2-[9-(3-hydroxy-2-methylbenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
3-methoxy-N-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]piperidine-1-carboxamide
methyl (2S)-1-[3-(3-cyclopentylpropanoyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]pyrrolidine-2-carboxylate
1-[3-(3-methylphenyl)phenyl]-N-(1H-1,2,4-triazol-5-ylmethyl)piperidin-4-amine
1-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
N-(cyclohexylmethyl)-1-[2-(3,4-dimethoxyphenyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
2-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
2-{2-[3-(dimethylamino)phenyl]phenoxy}propanamide
3-ethyl-8-(2-fluoro-6-methoxybenzoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 2-(diethylsulfamoyl)-6-(4,4,4-trifluorobutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-({3-[(2-chloro-4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-methyl-1H-pyrazol-5-amine
4-{1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}pyridine
(1S,6R)-9-(4-fluoro-3-hydroxybenzoyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
[2,4,6-trimethyl-3-({methyl[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenyl]methanol
3-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-5,6-dimethyl-1,2-dihydropyridin-2-one
2-(adamantan-1-yl)-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]acetamide
N,3-dimethyl-4-oxo-N-[3-(piperidin-1-yl)propyl]-3,4-dihydroquinazoline-7-carboxamide
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-ol
1-[2-(4-methylpentyl)morpholin-4-yl]pent-4-en-1-one
N-[(3S,4R)-1-(5-chloropyridin-2-yl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[4-(methylsulfanyl)benzoyl]pyrrolidin-3-yl]methanol
3-hydroxy-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]pyridine-2-carboxamide
N-(furan-3-ylmethyl)-N-methyl-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
(1R,5R)-6-[(2-methoxy-4-methylphenyl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(2S)-3-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propane-1,2-diol
1-(dimethyl-1,2-oxazole-4-carbonyl)-3-(3-fluorophenoxymethyl)piperidine
N-(2-methylphenyl)-3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
(3aR,6aS)-5-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(1-{1-[(2,3,4-trimethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N4-methylpyrimidine-2,4-diamine
1-[(2S)-2-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]pyrrolidin-1-yl]ethan-1-one
3-({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)propan-1-ol
1-[2-({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)ethyl]imidazolidin-2-one
methyl[(3-methylpyridin-4-yl)methyl]{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
5-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide