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2-[4-(1H-imidazol-1-yl)phenyl]-7-methyl-1H-1,3-benzodiazole
1-cyclopentyl-4-{[methyl({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]methyl}pyrrolidin-2-one
[1-(2-chlorobenzenesulfonyl)-4-[(4-methoxyphenyl)methyl]piperidin-4-yl]methanol
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,1-dimethyl-1H-indole-3-carboxamide
1-[(3-methoxyphenyl)methyl]-4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-2-one
1-{4-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-1-yl}-2-(phenylsulfanyl)ethan-1-one
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-3-(furan-2-yl)-N-methylpropanamide
2-phenyl-1-[3-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]ethan-1-one
N-cyclopropyl-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)methanesulfonamide
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-4-phenylbutane-1,4-dione
2-{1-[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]ethyl}phenol
(4aS,8aR)-1-(3-hydroxypropyl)-6-(quinolin-5-ylmethyl)-decahydro-1,6-naphthyridin-2-one
(1S,5R)-6-benzyl-3-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
8-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-{1-[(2-chlorophenyl)methyl]azepan-3-yl}-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-6-methoxy-1-methyl-1H-indole-2-carboxamide
1-[1-(3-cyclohexylpropanoyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
(2R,3R)-3-({[1-(2-hydroxyethyl)piperidin-4-yl]methyl}(methyl)amino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-({5-[(4-chloro-3-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
6-(3-chlorophenyl)-7-(3-methylbut-2-en-1-yl)-2-(pyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(4-methoxyphenyl)butanamide
N-{5-[(3S,4S)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-1,3-thiazol-2-yl}acetamide
3-{2-[ethyl({[5-(1H-pyrazol-3-yl)furan-2-yl]methyl})amino]-1-hydroxyethyl}phenol
(3S,4S)-1-[5-(hydroxymethyl)furan-2-carbonyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-(cyclopropylmethyl)-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)acetamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-(1-ethylpiperidin-4-yl)-N-[(4-methylphenyl)(pyridin-4-yl)methyl]acetamide
[(2,6-dichloro-3,4-dimethoxyphenyl)methyl](methyl)[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amine
N-(3-cyclopentylpropyl)-N,4-dimethylpentanamide
2-(3-methylthiophen-2-yl)-1-(3,4,5-trimethoxyphenyl)-1H-imidazole
1-[4-(4-phenyl-1H-imidazol-1-yl)phenyl]ethan-1-ol
2-methyl-N-{2-[7-(naphthalen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}propanamide
1-[(2,6-difluorophenyl)methyl]-4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidine
5-[(1,1-dioxo-1λ6-thian-4-yl)amino]-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-(2-aminoethyl)-4-[(1R)-1-(4-chlorophenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyridine
7,7-dimethyl-2-[(4-methyl-1,3-thiazol-5-yl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[(2-ethyl-4-methyl-1,3-oxazol-5-yl)formamido]hexanamide
(3aR,6aR)-2-[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(3-hydroxy-3-methylbutyl)-N-(1-phenylcyclopropyl)benzamide
(1S,5R)-3-[(4-methoxy-2-methylphenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
8-[(2E)-2-methylbut-2-en-1-yl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-ethylpiperazin-1-yl)-3-[2-methoxy-4-({[2-(2-methylphenyl)ethyl]amino}methyl)phenoxy]propan-2-ol
(2E)-N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]-3-(4-methoxyphenyl)prop-2-enamide
N-[1-(2-methoxyphenyl)propan-2-yl]-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)acetamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
1-{2-hydroxy-3-[2-methoxy-4-({methyl[3-(pyrrolidin-1-yl)propyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
(2S,4S)-4-amino-N,N-diethyl-1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}pyrrolidine-2-carboxamide
2-methoxyethyl 9-oxo-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxylate