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N-[(1-methylpiperidin-4-yl)methyl]-2-phenoxybenzamide
N-[(2-ethoxyphenyl)methyl]-4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
1-ethyl-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(4-{[2-(difluoromethoxy)phenyl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
{2-[4-(trifluoromethyl)pyrimidin-2-yl]phenyl}methanol
N-methyl-1-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)piperidine-3-carboxamide
1-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
N-(2-chloro-3,5-difluorophenyl)-3-(dimethylamino)pyrrolidine-1-carboxamide
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(pyridin-3-ylmethyl)propanamide
1-{7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(thiophen-2-yl)ethan-1-one
6-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]quinoxaline-5-carboxamide
methyl (2S)-1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)pyrrolidine-2-carboxylate
N-(1-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
[(3R,4R)-1-{[3-(2-aminoethyl)phenyl]methyl}-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-phenyl-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1,2,4-triazin-3-amine
3-[4-(2-cyclohexylpyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]-1-methylpyrrolidin-2-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-sulfamoylthiophene-2-carboxamide
3-methyl-5-propyl-N-[2-(pyridin-3-yl)ethyl]-1-benzofuran-2-carboxamide
N-(diphenylmethyl)-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
5-methyl-3-[1-(1H-pyrazol-1-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-amino-N-[(3R,4S)-4-cyclopropyl-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidin-3-yl]acetamide
N-cyclohexyl-N-cyclopropyl-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]pyrimidin-2-amine
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-fluoro-4-methylbenzamide
1-[1-(4,6-dimethylpyridine-3-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
4-fluoro-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)benzamide
3-(oxolan-3-yl)-5-(4-phenylphenyl)-1,2,4-oxadiazole
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-pyrazole-3-carboxamide
3-(dimethylamino)-1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
5-[1-(4-tert-butylbenzoyl)piperidin-4-yl]-5-[(2-chlorophenyl)methyl]imidazolidine-2,4-dione
N-[(2,3-dimethoxyphenyl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
2-(1-{[1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-(pyridin-2-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(2,3-difluorophenyl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
3-[1-(1,7-dimethyl-1H-indole-2-carbonyl)piperidin-3-yl]benzoic acid
N-[2-(7-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-(4-fluorophenyl)acetamide
4-(5-acetylthiophene-2-carbonyl)-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
5-chloro-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}thiophene-2-carboxamide
5-[3-(1H-pyrazol-3-yl)phenyl]furan-2-carboxamide
4,6-dimethyl-1-{2-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
4-[3-(benzyloxy)phenyl]-2-methyl-1H-imidazole
4-(1-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
9-{[3-(2-aminoethyl)phenyl]methyl}-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-1-(1-{[5-(methylcarbamoyl)furan-2-yl]methyl}piperidin-4-yl)piperidine-3-carboxamide
4-({2-[2-(pyridin-4-yl)-1H-imidazol-1-yl]phenyl}methyl)morpholine
5-[2-({3-azaspiro[5.5]undecan-9-yl}amino)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 4-(5-methyl-4-{[3-(thiophene-2-carbonyl)piperidin-1-yl]methyl}-1,3-oxazol-2-yl)benzoate
1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(propan-2-yl)-1H-1,3-benzodiazole