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2,5-dimethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
N3-[(3,4-difluorophenyl)methyl]-N5-(2-methoxyethyl)-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-{4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
4-(6-ethylpyrimidin-4-yl)-N-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)piperazine-1-carboxamide
2-[1-(2-methoxyphenyl)-5-[(propan-2-yloxy)methyl]-1H-1,2,4-triazol-3-yl]acetamide
1-(1-benzyl-1H-pyrazole-4-carbonyl)-3-(1H-imidazol-2-yl)piperidine
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]cyclopentanamine
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl){[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}amine
N-methyl-2-oxo-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]propanamide
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2-(propan-2-yloxy)ethyl]benzamide
2-[5-(2H-1,3-benzodioxol-5-yl)-1H-indol-1-yl]-N-(1,3-dimethyl-1H-pyrazol-5-yl)acetamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)benzamide
5-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(1S,6R)-3-[(8-methoxy-2H-chromen-3-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-ethyl-N-(2-methylprop-2-en-1-yl)acetamide
2-[1-(2-methoxyethyl)piperidine-4-carbonyl]-6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline
2-({[2-(4-chlorophenyl)ethyl]amino}methyl)-4-(6-methoxypyridin-2-yl)phenol
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-methyl-6-[2-(phenylsulfanyl)acetyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-[(2,6-difluorophenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(azepane-1-carbonyl)-1-ethyl-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(carbamoylamino)-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)acetamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
1-(2-{[3-(pyridin-4-yl)propyl]amino}pyrimidin-4-yl)piperidin-3-ol
4-(1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)morpholine
3-(2-chlorophenyl)-3-{2-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-1-methylpyrrolidine-2,5-dione
2-amino-1-{6-methyl-5-[5-(oxan-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}ethan-1-one
3-(azepane-1-carbonyl)-1-(prop-2-en-1-yl)-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-5-[(methylsulfanyl)methyl]furan-2-carboxamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1-[(diethylcarbamoyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-1-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
9-[2-(methylamino)-1,3-thiazole-4-carbonyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(1-{[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[2-(4-{[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
2-[3-(2-fluorophenyl)-1H-pyrazol-1-yl]-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
2-[1-benzyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[1-(thiophen-2-yl)ethyl]acetamide
N-[(3R,4S)-4-cyclopropyl-1-(3-hydroxypropyl)pyrrolidin-3-yl]-1-(2-fluorophenyl)cyclopropane-1-carboxamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(pyridin-3-yloxy)propyl]acetamide
(2,1,3-benzoxadiazol-5-ylmethyl)({[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl})amine
(7S,8aS)-7-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-{2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}azepane
5,7-dimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
(2R,4S)-1-(1,3-benzothiazole-6-carbonyl)-4-hydroxypiperidine-2-carboxylic acid
N,N-dimethyl-2-[(1S,5R)-6-(1-methyl-1H-indole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
[(2S,4R,5R)-4-[({[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}amino)methyl]-5-(2-fluorophenyl)-1-methylpyrrolidin-2-yl]methanol
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-(1-methoxybutan-2-yl)pyridin-2-amine
4-(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)thiomorpholine
2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[(5-methylthiophen-2-yl)methyl]acetamide
2-[methyl(2-phenylethyl)amino]-N-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-indene-2-carboxamide
2-(3-methoxyphenoxymethyl)-4-(pyrrolidine-1-carbonyl)-1,3-oxazole