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1-benzyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-3-amine
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-oxo-N-phenylacetamide
2-(4-{2-[2-(4-methoxyphenyl)-1H-imidazol-1-yl]ethyl}piperazin-1-yl)pyrimidine
2-(4-{[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol
1-[(2,3-dimethoxyphenyl)methyl]-3-[4-(methylsulfanyl)benzoyl]piperidine
(3S,9aR)-3-benzyl-8-[(3,4-difluorophenyl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-1-(pyrrolidin-1-yl)cyclohexane-1-carboxamide
2,4-difluoro-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]benzamide
[(2,3-dimethyl-1H-indol-5-yl)methyl][1-(pyridin-3-yl)propan-2-yl]amine
5-oxo-N-[2-(pyridin-3-yl)ethyl]-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyridin-4-yl)piperazine
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(methoxymethyl)piperidine
N-benzyl-3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxamide
2-[4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-1-yl]pyrimidine
1-({1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
3-(2-ethoxyphenyl)-1-(1,4-oxazepan-6-ylmethyl)urea
4-{[2-(benzyloxy)phenyl]methyl}piperazine-1-sulfonamide
1-(cyclopropylmethyl)-3-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
1-(8-chloro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-methylurea
methyl (2S)-1-({4-[(2,3-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)pyrrolidine-2-carboxylate
4-(1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine-3-carbonyl)morpholine
2-{4-[6-amino-2-(diethylamino)pyrimidin-4-yl]piperazin-1-yl}ethan-1-ol
(3R,4R)-3-cyclobutyl-4-methyl-1-(1-methyl-4-phenylpiperidine-4-carbonyl)pyrrolidin-3-ol
2-{[(1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-chloropyridin-2-yl)piperidin-3-ol
1-(1-methylpiperidin-4-yl)-N-(2-phenylpropan-2-yl)piperidine-3-carboxamide
1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
2-chloro-N-(2-{[2-(4H-1,2,4-triazol-4-yl)pyridin-4-yl]formamido}ethyl)benzamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2-(trifluoromethyl)-1H-1,3-benzodiazole
N-[2-(3,5-dimethoxyphenyl)ethyl]-2-methylpyrimidine-5-carboxamide
N-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-3-(thiophene-2-carbonyl)piperidine-1-carboxamide
5-(1-benzofuran-2-yl)-N-[3-(1H-pyrazol-1-yl)propyl]-1,2,4-triazin-3-amine
3-fluoro-5-{4-[(4-methoxyphenyl)methyl]-3-oxopiperazine-1-carbonyl}benzonitrile
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-(1H-imidazol-2-ylmethyl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
4-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-1-methylpiperazin-2-one
1-(4-methyl-1H-pyrrole-2-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
(3S,4S)-1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
2-(3-fluorophenoxymethyl)-N-[1-(3-methylpyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
1-[(1-cyclohexyl-1H-1,2,4-triazol-5-yl)methyl]-1,4-dihydroquinolin-4-one
1-ethyl-N-[2-(4-methoxyphenyl)ethyl]-3-(4-methylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl 3-({3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}amino)propanoate
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}-1-(furan-3-carbonyl)piperidine
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylacetamide
methyl (2R,4S)-1-(2,8-dimethylquinoline-3-carbonyl)-4-hydroxypiperidine-2-carboxylate
1-[1-(4-{[(3-methoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperidin-4-yl]piperidin-3-ol
6-ethyl-4-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-2H-chromen-2-one
ethyl 2-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-1,3-oxazole-4-carboxylate
10-methoxy-5-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
3,5,7-trimethyl-2-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]-1H-indole