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{5-[(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)methyl]furan-2-yl}methanol
1-(2-phenylethyl)-2-(propane-2-sulfonyl)-5-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}-1H-imidazole
8-methoxy-5-{7-methylthieno[3,2-d]pyrimidin-4-yl}quinoline
2-chloro-4-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}phenol
N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-thiazole-5-carboxamide
(1R,5R)-6-(cyclopropylmethyl)-N-(2,5-dimethoxyphenyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-[4-(4-phenyl-1H-imidazol-5-yl)phenyl]-2H-1,2,3,4-tetrazole
3-tert-butyl-1-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]urea
(2S)-2-[4-(2,4-difluoro-3-methoxyphenyl)-1H-1,2,3-triazol-1-yl]-4-methylpentanamide
2-(5-acetylthiophen-3-yl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)furan-2-carboxamide
4-(pyrazin-2-yl)-2-({4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}methyl)phenol
2-{4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-3-(pyrrolidin-1-yl)piperidine
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
2-amino-4-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
3-(1H-pyrazol-1-ylmethyl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
3-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}-1,2-dihydroquinoxalin-2-one
9-(2-methyl-1H-pyrrole-3-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-3-ol
ethyl({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})(pyridin-4-ylmethyl)amine
1-(4-chloro-2-fluorobenzoyl)-N-(3-fluorophenyl)piperidin-3-amine
1-methyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-3-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
methyl 3-[(3S,4R)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoate
3-amino-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}thiophene-2-carboxamide
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-[5-methoxy-2-({[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
4-ethyl-3-{1-[(4-methanesulfonylphenyl)methyl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(3-methylthiophene-2-carbonyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine
2-{1-[(4-fluorophenyl)methyl]-4-{4-[(propan-2-yl)amino]pyrimidin-2-yl}piperazin-2-yl}ethan-1-ol
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-(4-phenylpiperidin-1-yl)butan-1-one
3-oxo-N,N-bis(propan-2-yl)-2,8-diazaspiro[4.5]decane-8-carboxamide
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]propanamide
8-[(3S,4S)-1-(1-benzothiophen-2-ylmethyl)-4-hydroxypyrrolidin-3-yl]-2-methyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
2-[(2-hydroxyethyl)({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propan-1-one
4-[4-(2-ethoxyethyl)piperazin-1-yl]-5-ethylpyrimidin-2-amine
2-cyclopropyl-N-[2-(piperidin-1-yl)ethyl]-1,3-benzoxazole-6-carboxamide
4-({methyl[2-(oxan-2-yl)ethyl]amino}methyl)benzonitrile
N-[3-({[2-(furan-2-ylmethyl)-3-hydroxypropyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
4-methyl-5-{2-[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]ethyl}-1,3-thiazole
N-(2-acetamidophenyl)-2-[(2-methanesulfonamidoethyl)amino]acetamide
3-(1,3-dimethyl-1H-pyrazol-5-yl)-4-[2-(4-fluorophenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aR,7aS)-1-{2-[4-(1H-1,2,4-triazol-1-yl)phenoxy]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[4-(2-phenoxypropanoyl)piperazin-1-yl]-2-(pyridin-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
{4-[1-(2-phenylethyl)piperidin-4-yl]-1,4-oxazepan-6-yl}methanol
2-[(2-{[1-(2,6-dimethylphenoxy)propan-2-yl]carbamoyl}phenyl)amino]acetic acid