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1-ethyl-5-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
1-(2-methoxyphenyl)-2,2-dimethyl-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazine
5-oxo-1-(pyridin-4-ylmethyl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}pyrrolidine-3-carboxamide
3-[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]phenol
2-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}acetamide
4-{1-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}benzoic acid
2-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
5-[(3,4-difluorophenyl)methyl]-4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-cyclohexyl-4-[2-(pyridin-2-ylsulfanyl)acetyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
5-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
2-(2-cyclopropylacetyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-(4-cyano-2,5-difluorophenyl)-3-methylurea
1-(furan-2-ylmethyl)-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]piperidine-4-carboxamide
1-[(4-fluorophenyl)methyl]-4-(5-fluoropyridine-2-carbonyl)-2-(propan-2-yl)-1,4-diazepane
5-cyclopropyl-N-[2-(diethylamino)ethyl]-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
9-(3-ethyl-1,2-oxazole-5-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
2-chloro-5-(4-methoxy-3-methylphenyl)pyrazine
1-[2-hydroxy-3-(4-methoxy-2-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)propyl]piperidin-4-ol
2-(4-methylpentyl)-4-{4H-thieno[3,2-b]pyrrole-5-carbonyl}morpholine
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-2-ylmethyl)acetamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanamide
5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)-5-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}imidazolidine-2,4-dione
N-(4-carbamoyl-2-methylphenyl)-4-[2-(methylsulfanyl)ethyl]piperazine-1-carboxamide
{2-[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]ethyl}dimethylamine
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
N-[(2,3-difluorophenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
benzyl N-[1-(6-ethylpyrimidin-4-yl)pyrrolidin-3-yl]carbamate
1'-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
2-(3-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1H-pyrazol-3-yl}phenyl)-4-(trifluoromethyl)pyrimidine
{4-[(2-chlorophenyl)methyl]-1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-yl}methanol
(2S)-2-{[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}-4-(methylsulfanyl)butan-1-ol
4-methyl-6-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-1,3-benzothiazol-2-amine
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(1-ethyl-1H-pyrazol-4-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
5-[4-(2-methylphenoxy)piperidine-1-carbonyl]-2-(pyridin-2-yl)pyrimidine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-2-methoxy-N-(oxolan-2-ylmethyl)benzamide
(1-{[4-(5-methylfuran-2-yl)phenyl]methyl}piperidin-3-yl)methanol
4-{1-azabicyclo[3.2.1]octan-5-yloxy}-3-methoxybenzonitrile
9-(3,4-difluorophenyl)-15-methyl-13-oxo-N-(pyridin-2-ylmethyl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
methyl (2S)-2-[(4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}phenyl)formamido]-3-methylbutanoate
[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]methanesulfonamide
[(2S)-1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidin-2-yl]methanol
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-methyl-1H-indol-1-yl)ethyl]acetamide
N-ethyl-2-(3-methylpentanamido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
2-methoxy-N-[(2R,3R)-2-(prop-2-en-1-yloxy)-1'-(1,3-thiazol-2-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(quinolin-2-yl)piperidin-3-ol
1-(2,3-dihydro-1H-indene-1-carbonyl)-4-(2-methoxybenzoyl)piperazine
2-(2,3-dihydro-1H-inden-1-yl)-1-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)ethan-1-one