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(4aR,8aR)-1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-6-(3-methoxybenzoyl)-decahydro-1,6-naphthyridine
(3S,4S)-1-{[2-(benzylamino)pyrimidin-5-yl]methyl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
4-[2-(5-methylpyridin-3-yl)pyridine-4-carbonyl]morpholine
2-(3-chlorophenyl)-N-[4-(4-{[(3-methoxyphenyl)methyl]amino}piperidin-1-yl)phenyl]acetamide
(3S,4R)-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
2-[2-(3-chloro-2,4-difluorophenyl)-1H-imidazol-1-yl]-N-methylpentanamide
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}propane-1,2-dione
N-[(2-methoxyphenyl)methyl]-2-{methyl[1-(1,3-thiazol-2-yl)ethyl]amino}acetamide
5-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
N-[1-({[(4-phenyl-1,3-thiazol-5-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
2-chloro-4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
1-{[4-(difluoromethoxy)phenyl]methyl}-N-(4-fluorophenyl)piperidin-3-amine
3-methoxy-1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}propan-1-one
N-[(3S,4R)-4-propyl-1-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-3-yl]acetamide
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butan-1-one
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]pyridin-2-amine
methyl 2-{[5-(4-fluorophenyl)-4-(1-propanoylpiperidin-3-yl)pyrimidin-2-yl]sulfanyl}acetate
1-(2-methoxyethyl)-6-oxo-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide
N-(4-ethylphenyl)-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
2-acetyl-8-{[4-(2-methylpropyl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-[(2-methylphenyl)methyl]-1-(quinolin-2-yl)piperidine-3-carboxylic acid
(3R,4R)-4-cyclobutyl-3-methyl-1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]piperidin-4-ol
2-(furan-3-carbonyl)-1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
N-butyl-N-[(2-methylphenyl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
methyl 3-{[4-(5-methylthiophene-2-carbonyl)-7-oxo-1,4-diazepan-1-yl]methyl}benzoate
5-oxo-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
N-(2-methylpropyl)-1-[1-(2-phenoxyacetyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
5-[(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-N,N-dimethylpyridin-2-amine
1-(1-benzofuran-5-ylmethyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
(3R,4R)-4-(azepan-1-yl)-1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-ol
N-{3-[(5-methylpyridin-2-yl)amino]propyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
6-(cyclopropylmethoxy)-4-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-1-[(3-methoxyphenyl)methyl]-1,4-diazepan-2-one
4-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyrimidine
7-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-{5-[(4aR,8aR)-6-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-decahydro-1,6-naphthyridine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
1-(3-methoxyphenyl)-2,2-dimethyl-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1,2,5-trimethyl-N-(pyridin-4-ylmethyl)-1H-pyrrole-3-carboxamide
4-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-6-(propan-2-yl)-2-(trifluoromethyl)pyrimidine
N-{1-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-4-yl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
2-amino-4-[2-(2-methoxyethyl)pyrimidin-5-yl]-5H,6H,7H-pyrrolo[2,3-h]quinoline-3-carbonitrile
(2S,4R)-4-(4-{2-[(2-chlorophenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
1-{5-[(2H-1,3-benzodioxol-5-yl)carbamoyl]furan-2-yl}-1H-imidazole-4-carboxylic acid
5-(1,2-oxazolidine-2-carbonyl)-1-(2-phenylethyl)piperidin-2-one
1-(carbamoylmethyl)-N-{1-[(3-methylphenyl)methyl]cyclopropyl}piperidine-4-carboxamide
N-[2-(4-benzylpiperazin-1-yl)ethyl]-5,6-dimethylpyrimidin-4-amine
3-(4-fluoropiperidine-1-carbonyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine
2-{1-[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]piperidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
N-[(3S,4R)-1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide