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6-{[1-(hydroxymethyl)cyclopentyl]methyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
6-chloro-2-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}quinoline
8-(4-chloro-2-methoxybenzoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-methyl-5-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-3,4-dihydropyrimidin-4-one
2-(dimethylamino)-N-[2-methyl-5-(4H-1,2,4-triazol-4-yl)phenyl]acetamide
(1R,5R)-3-(2-ethoxybenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
3-(3-fluoro-4-phenylbenzoyl)-1-(furan-2-carbonyl)piperidine
3-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}methyl)-N,N-dimethyl-1,2,4-oxadiazole-5-carboxamide
{[5-(furan-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}(methyl)[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-methyl-N-(2-phenylethyl)-1-(pyridin-3-ylmethyl)piperidin-3-amine
N,N,7,8-tetramethyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
N-(cyclohexylmethyl)-5-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
2-(adamantan-1-yl)-4-hydroxy-N-methyl-N-[2-(methylamino)ethyl]pyrimidine-5-carboxamide
2-acetyl-8-(2-phenylethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(4-methyl-1,3-thiazol-2-yl)-2-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoacetamide
N-cyclohexyl-4-{2-methylimidazo[1,2-a]pyrimidine-3-amido}piperidine-1-carboxamide
1-{4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-(4-{[(3S,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
3-methyl-4-(6-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-1-[(3-methylphenyl)methyl]piperazin-2-one
2-(ethylamino)-N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}pyrimidine-5-carboxamide
dimethyl(2-{[(2-methylphenyl)methyl][(2-propylpyrimidin-5-yl)methyl]amino}ethyl)amine
4-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carboxylic acid
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}({[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
(3S,4R)-1-[(5-fluoro-2-methoxyphenyl)methyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
2-[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-hydroxy-1-(2-phenylethyl)-3-{[(thiophen-2-ylmethyl)amino]methyl}piperidin-2-one
5-(1-benzylpiperidin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
N-cyclooctyl-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]-N-propylacetamide
1-{1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]azetidin-3-yl}-2-methylpiperidine
(4aS,8aR)-6-(2-chloro-4-fluorobenzoyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-4-(piperidin-3-yl)benzamide
2-ethyl-N,4-dimethyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-1,3-thiazole-5-carboxamide
N-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-2,3-dihydro-1H-inden-2-amine
(1S,3R)-3-[3-(5-methyl-1H-pyrazol-1-yl)propanamido]-N-(thiophen-2-ylmethyl)cyclopentane-1-carboxamide
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-4-(1H-pyrazol-3-yl)piperidine-1-carboxamide
2-chloro-5-acetamido-N-[(5-methoxy-1H-indol-2-yl)methyl]benzamide
6-(3-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}piperidin-1-yl)pyridine-3-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[3-(morpholin-4-yl)propyl]benzamide
4-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)acetamide
4-(4-methoxy-4-phenylpiperidin-1-yl)-6-methylpyrimidin-2-amine
2-hydroxy-N-(isoquinolin-5-ylmethyl)-N-methyl-4-(methylsulfanyl)butanamide
3-methanesulfonyl-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
4-(2,1,3-benzothiadiazol-4-yl)-3-tert-butyl-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(2S,5R)-1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)-2,5-dimethylpiperazine