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2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]acetamide
4-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
7-(3-chloro-5-methoxybenzoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(trifluoromethyl)pyrimidin-4-amine
2-(3-fluorophenoxymethyl)-N-methyl-N-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
methyl 3-({[4-(2-methylpropoxy)phenyl]methyl}(pyridin-4-ylmethyl)sulfamoyl)thiophene-2-carboxylate
[2-({4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
(1R,2S,9R)-11-(quinolin-4-ylmethyl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
9-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(6-phenylpyridazin-3-yl)piperidin-3-ol
3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-5,6,7,8-tetrahydroquinoline
N-(3-carbamoylphenyl)-4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carboxamide
2-[2-methyl-3-({[3-(pyridin-3-yloxy)propyl]amino}methyl)-1H-indol-1-yl]acetamide
2-(4-fluorophenyl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
(3S,4S)-1-(3-methylthiophene-2-carbonyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-{[5-(1H-1,2,4-triazol-5-ylsulfanyl)furan-2-yl]methyl}piperidine
4-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}morpholine
(1R,3s,6r,8S)-4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-azatricyclo[4.3.1.13,8]undecane
[(3R,4R)-4-[(dimethylamino)methyl]-1-(2-propoxybenzoyl)pyrrolidin-3-yl]methanol
1-(1,2-oxazol-3-ylmethyl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-(1-{7-[(2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)oxolane-3-carboxamide
1-(2-methylpropyl)-5-[1-(prop-2-en-1-yl)pyrrolidine-2-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
N-methyl-6-(4-propylpiperazin-1-yl)-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
3-(1H-1,3-benzodiazol-2-yl)-1-[4-(pyridin-4-yl)piperidin-1-yl]propan-1-one
3-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-1-[4-(oxan-2-ylmethoxy)phenyl]urea
3-(benzyloxy)-1-(1H-1,2,3-triazole-5-carbonyl)piperidine
N4-methyl-N2-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)pyrimidine-2,4-diamine
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
methyl 3-[(3-methylphenyl)methyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
4-phenyl-5-[2-(prop-2-en-1-yloxy)phenyl]-1-[2-(1H-pyrazol-4-yl)ethyl]-1H-imidazole
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
8-(4-phenyl-1,3-thiazol-2-yl)-2,8-diazaspiro[4.5]decan-3-one
N-(furan-2-ylmethyl)-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2-[methyl(piperidin-4-yl)amino]acetamide
methyl 9-[2-(2-fluorophenyl)ethoxy]-3-{[5-(hydroxymethyl)furan-2-yl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-ethyl-2-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyrimidine
1-(pyridin-2-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-(3-ethylphenyl)-N'-[(5-ethylpyridin-2-yl)methyl]butanediamide
N-{1-oxaspiro[4.4]nonan-3-yl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
3-methyl-8-(3-methyl-2-phenylbutanoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-2-phenylethyl}(2-methoxyethyl)(pyridin-3-ylmethyl)amine
1-[4-({2-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]phenyl}methyl)piperazin-1-yl]ethan-1-one
1-[6-methyl-2-(methylamino)pyrimidin-4-yl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N-(1-{[6-(dimethylamino)pyridin-3-yl]methyl}piperidin-4-yl)methanesulfonamide
N-(3-methoxyphenyl)-2-{4-[3-(4H-1,2,4-triazol-4-yl)propanoyl]morpholin-3-yl}acetamide
5-(2,6-difluorophenoxymethyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
ethyl 3-({3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carbonyl}amino)propanoate