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(4aS,8aR)-6-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-(3-methylcinnolin-5-yl)-3-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}urea
4-methyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2-(methylamino)-1,3-thiazole-5-carboxamide
N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
5-(3-fluoro-4-methoxyphenyl)-N-[(6-methylpyridin-2-yl)methyl]-1,2,4-triazin-3-amine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-{[(methylcarbamoyl)methyl]amino}pyridine-3-carboxamide
2-(4-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperazin-1-yl)pyrimidine
N-[(1-propylcyclobutyl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-hydroxy-3-({[(5-methylthiophen-2-yl)methyl]amino}methyl)-1-(2-phenylethyl)piperidin-2-one
3,3-dimethyl-1-[(5-{[4-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea
1-{3-oxo-3-[3-(2-phenylacetyl)piperidin-1-yl]propyl}azepan-2-one
4-methyl-6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-2-amine
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidine
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-2-(2-oxopiperidin-1-yl)acetamide
2-[(3,4-dimethoxyphenyl)methyl]-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
methyl 2-{[4-(1-acetylpiperidin-3-yl)-5-(4-fluorophenyl)pyrimidin-2-yl]sulfanyl}acetate
3-{[(1,3-benzothiazol-2-ylmethyl)amino]methyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
2-{3-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenoxy}acetamide
3-propyl-4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazole
1-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-4-carboxamide
1-methyl-5-[3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-1H-1,2,3-benzotriazole
1-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
methyl 3-{[4-(dimethylamino)phenyl]methyl}-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-ethyl-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(2-methylprop-2-en-1-yl)propanamide
methyl 1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidine-2-carboxylate
1-cyclopentyl-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
2-(2-methoxyethoxy)-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
N-butyl-4-{3-[(pyridin-2-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxamide
(1S,5R)-6-(3-fluoro-4-methoxybenzoyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[4-({[2-(cyclohex-1-en-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(diethylamino)propan-2-ol
2-amino-7-[2-(oxan-2-ylmethoxy)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-1,2-oxazole-3-carboxamide
2-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(phenylsulfanyl)acetamide
5-(4-fluorophenyl)-N-(3-phenylpropyl)-1,2,4-triazin-3-amine
2-{benzyl[1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}ethan-1-ol
methyl N-{2-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]-2-oxoethyl}carbamate
1-{2-oxo-2-[4-(4-phenylpyrimidin-2-yl)piperazin-1-yl]ethyl}-1,2-dihydropyrimidin-2-one
3-{1-[3-(furan-2-yl)benzoyl]piperidin-3-yl}-N-[(3-methoxyphenyl)methyl]propanamide
4-(pyrazin-2-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-1-benzothiophene-2-carboxamide
1-methyl-4-{[4-(2-methylphenyl)phenyl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-(4-chlorophenyl)ethyl]-1-cycloheptyl-6-oxopiperidine-3-carboxamide
N-{3-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-oxopropyl}-N-methylmethanesulfonamide
3-fluoro-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyridin-2-amine
1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-[4-(1H-pyrazol-1-yl)butan-2-yl]urea
3-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}methanesulfonamide
5-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}-N,N,4-trimethylpyrimidin-2-amine