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(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amine
N-(2-chlorophenyl)-3-[1-(4,4,4-trifluorobutyl)piperidin-4-yl]propanamide
6-(6-fluoroquinolin-8-yl)-2-(pyrrolidin-1-yl)pyrimidin-4-amine
2-amino-5-ethyl-4-[5-(hydroxymethyl)furan-2-yl]-6-phenylpyridine-3-carbonitrile
2-({1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)quinolin-8-ol
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
(3aS,6aS)-2-[(3-methyl-1,2-oxazol-5-yl)methyl]-5-(1-methyl-1H-pyrrole-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{2-[3-(benzyloxy)azetidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,2-benzothiazol-3-one
N-(4-fluoro-2-methylphenyl)-2-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}formamido)acetamide
5-(2,6-difluorophenoxymethyl)-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
methyl 3-{[1-(cyclopropylmethyl)-5-(naphthalene-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
N-(1-carbamoylcyclopentyl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
6-(4-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidine-1-carbonyl)-1H-indole
3-(3-methoxyphenyl)-5-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propyl}-1,2,4-oxadiazole
N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-5-fluoro-N,N-dimethylpyrimidin-4-amine
N-[2-(dimethylsulfamoyl)ethyl]-3-(4-methoxyphenyl)-3-phenylpropanamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)butane-1-sulfonamide
2-{8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
9-{2-[4-(hydroxymethyl)phenyl]acetyl}-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}-5-methylpiperidin-2-one
(2-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)urea
methyl 5-[3-(furan-2-yl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]-2-hydroxybenzoate
3-chloro-N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]benzamide
4-methyl-3-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
5-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
methyl 3-[(3,4-difluorophenyl)methyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-3,4-dihydrophthalazine-1-carboxamide
N-(isoquinolin-5-ylmethyl)-N-methyl-2H-1,3-benzodioxole-5-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
N-[2-(propan-2-yloxy)ethyl]-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
6-(3-fluorophenyl)-N-(2-hydroxyethyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[3-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)propyl]acetamide
9-[(3-fluoro-5-methylphenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[4-(hydroxymethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
8-(3-methylpyridin-2-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 5-{[(2E)-3-(furan-2-yl)prop-2-en-1-yl]amino}-1-(2-methoxyethyl)-3-(3-methylbutanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}-1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidine
methyl 4-[4-(4-methyl-1,3-thiazol-2-yl)piperazin-1-yl]benzoate
3-chloro-N-cyclopentyl-N-({4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)benzamide
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-2-(morpholin-4-yl)-6-phenylpyridine-3-carboxamide
2-(5-methoxyfuran-2-carbonyl)-1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
6-ethyl-N-{[1-(methoxymethyl)cyclopentyl]methyl}pyrimidin-4-amine
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperazine
2-(cyclopropylmethyl)-9-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{2-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-chlorophenyl)urea
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-4-(1H-1,2,4-triazol-1-yl)butanamide
N-(1H-indol-5-ylmethyl)-2-(methylamino)pyridine-4-carboxamide
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-(quinolin-4-ylmethyl)pyrrolidin-3-yl]methanol