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(2S)-2-amino-N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)butanamide
(1S,3R)-3-amino-N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}cyclopentane-1-carboxamide
5-[2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-(4-acetylphenoxy)-1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
1-(4-methylphenyl)-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazin-2-one
(4aR,7aS)-1-[(2-methylphenyl)methyl]-4-(pyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{3-benzyl-1-[(2-chloro-4-fluorophenyl)methyl]piperidin-3-yl}methanol
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
(3S,4S)-1-[(4-methoxy-3-methylphenyl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
4-({[(3-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]amino}methyl)hepta-1,6-dien-4-ol
N3-[(5-chlorothiophen-2-yl)methyl]-N5-ethyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
methyl[(4-phenoxyphenyl)methyl]{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
4-(cyclopropylmethyl)-1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
3-(3-cyclohexyl-1H-1,2,4-triazol-5-yl)-1-[(5-fluoro-1H-indol-2-yl)methyl]-1-methylurea
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(furan-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4,5-dimethyl-6-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
8-(2,2-dimethyloxane-4-carbonyl)-2-(3-methylbutyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-{4-[1-(2,1,3-benzoxadiazol-5-ylmethyl)pyrrolidin-3-yl]pyridin-2-yl}phenol
(2S,4R)-4-{[(3,4-difluorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
2-[1-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
diethyl({[3-(3-ethylpiperazine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
7-{1-ethyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}-1,2,3,4-tetrahydroquinoxalin-2-one
1-(4-{1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-carbonyl}-3,5-dimethyl-1H-pyrrol-2-yl)ethan-1-one
3-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propanoic acid
2-(4-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}piperazin-1-yl)-5-methyl-1,3-benzoxazole
methyl({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
8-(1-benzothiophen-2-ylmethyl)-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-chloro-4-fluoro-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1-benzothiophene-2-carboxamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-methoxynaphthalen-1-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-{1-[2-chloro-5-(trifluoromethyl)benzoyl]piperidin-4-yl}-N-cyclopropylpropanamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-[(2-methoxyphenyl)methyl]-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
3-[1-(1-benzyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
N-cyclopropyl-2-(cyclopropylmethyl)-7-(1H-imidazol-4-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]oxane-2-carboxamide
2-methyl-2-[4-(morpholin-4-yl)-2-{[1-(pyridin-3-yl)propan-2-yl]amino}pyrimidin-5-yl]propanoic acid
3-[5-({methyl[3-(phenylsulfanyl)propyl]amino}methyl)thiophen-3-yl]prop-2-yn-1-ol
(3S,4S)-1-cyclobutanecarbonyl-4-[4-(pyrazin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
2-(2-{1-[2-(2-oxoazepan-1-yl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
(3-{2-[1-(1,3-benzoxazol-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
(1R,5R)-6-(cyclobutylmethyl)-3-(2,3-difluoro-4-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
1-(cyclohexylmethyl)-N5-ethyl-N3-methyl-4-oxo-N3-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
N'-(2,4-dimethylphenyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}propanediamide
1-{4-[2-(2,2-diphenylethyl)morpholin-4-yl]piperidin-1-yl}ethan-1-one
4-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-N-(3-hydroxyphenyl)-4-oxobutanamide
N-[2-(dimethylamino)ethyl]-3-{1-[(2,4,5-trimethylphenyl)methyl]piperidin-4-yl}propanamide
3-(4-methoxy-3,5-dimethylbenzoyl)-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidine
(3R)-N-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-amine