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N-[(4-hydroxyphenyl)methyl]-3-(propan-2-yl)-N-(pyridin-4-ylmethyl)-1,2-oxazole-5-carboxamide
{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}(pyridin-2-ylmethyl)amine
5-[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
2-[1-(3-methylbutyl)-4-[1-(2-phenylethyl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
1-phenyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]spiro[2.4]heptane-1-carboxamide
N-methyl-1-(pyrazine-2-carbonyl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-amine
1-(4-benzylpiperazin-1-yl)-3-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]propan-1-one
(1R,7S)-6-(morpholine-4-carbonyl)-3-[2-(piperidin-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
6-{2-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
(3S,4S)-3-hydroxy-4-{2-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}-1λ6-thiolane-1,1-dione
4-(2-amino-6-methylpyrimidin-4-yl)-1-cyclopentylpiperazin-2-one
1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
7-(2-methoxyacetamido)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-4-methylpyrimidine-5-carboxamide
1-(2-{[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]amino}-4-methylpyrimidin-5-yl)ethan-1-one
1-cyclopentyl-N-[(1-hydroxycyclohexyl)methyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
8-(1-hydroxypropan-2-yl)-1-(2-methoxyethyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(2-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}ethyl)-1λ6-thiolane-1,1-dione
ethyl 4-{[5-(2,5-dimethylfuran-3-yl)-1,2,4-triazin-3-yl]amino}piperidine-1-carboxylate
2-(1H-indol-3-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2,6-dimethylpyridine
ethyl[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(2-chlorophenyl)methyl]-3-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}propanamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
N-ethyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-sulfamoylbenzamide
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
(1S,2R)-2-({[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}(methyl)amino)cyclohexan-1-ol
5-[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(furan-2-yl)ethane-1,2-dione
dimethyl[2-(2-{1-[6-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}-1H-imidazol-1-yl)ethyl]amine
9-[(2-chloro-3,4-dimethoxyphenyl)methyl]-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
3-[5-(4-chloro-2-methylphenoxymethyl)-3-methyl-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-[4-(trifluoromethyl)phenyl]ethan-1-one
3-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2-{[(2-fluorophenyl)methyl]sulfanyl}phenyl)pyridazine-4-carboxamide
(3R,4R)-1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
3-chloro-N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]benzamide
[(3S,5R)-1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
2-[2-(2,3-dihydro-1H-indol-1-yl)-2-oxoethyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-[2-methyl-2-(1H-pyrrol-1-yl)propanoyl]-4-phenoxypiperidine-4-carboxylic acid
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(pyridin-4-ylsulfanyl)acetamide
3-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
2-{3-[2-(methylsulfanyl)ethyl]-5-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-1,2,4-triazol-1-yl}acetic acid
{3-ethyl-1-[4-(4-methylpiperazin-1-yl)benzoyl]piperidin-3-yl}methanol
N,N-dimethyl-2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetamide
5-[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-3-propyl-1,2,4-oxadiazole
2-methyl-4-(4-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}phenyl)butan-2-ol
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
8-chloro-3-(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)-[1,2,4]triazolo[4,3-a]pyridine