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3-[(1-ethylcyclobutyl)methyl]-1-(1-methyl-1H-1,2,4-triazol-3-yl)urea
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-3-(1H-pyrazol-4-yl)propan-1-one
3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
methyl 4-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]benzoate
methyl 4-[ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)carbamoyl]butanoate
(4aR,7aS)-1-benzyl-4-{2-[ethyl(methyl)amino]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(1H-imidazol-1-ylmethyl)-1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-4-ol
7-(3-chlorophenyl)-4-(quinolin-8-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-{[(3R,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
3-{[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}-4-[(5-methylfuran-2-yl)methyl]piperazin-2-one
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
(3R,4R)-3-cyclobutyl-1-(4-methoxybenzenesulfonyl)-4-methylpyrrolidin-3-ol
N-methyl-N-[3-(morpholin-4-yl)propyl]-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[1-(thiophen-3-yl)propan-2-yl]acetamide
N-[1-(pyridin-2-yl)propan-2-yl]-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
(1S,5R)-3-{[3-(3,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonane
6-{[2-(dimethylamino)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
4-(1H-pyrazol-4-yl)-N-{1-[2-(trifluoromethyl)phenyl]ethyl}butanamide
1-(2-fluorobenzoyl)-3-(4-fluorophenoxymethyl)piperidine
2-methyl-N-[1-(3,4,5-trimethoxyphenyl)ethyl]-1-benzofuran-5-carboxamide
N-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-N-methylcyclohexanamine
6-methyl-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
2-[4-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazole-5-carbonyl)morpholin-3-yl]-N-(pyridin-3-yl)acetamide
N-(2,3-dihydro-1H-inden-2-yl)-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
3-{4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}propane-1,2-diol
N-[2-(azepan-1-yl)ethyl]-N-methyl-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
(1R,5R)-3-cyclobutanecarbonyl-6-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrrolidine-1-carboxamide
6-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,3-benzothiazol-2-amine
1-[3-(4-methylphenoxymethyl)piperidin-1-yl]-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}ethan-1-one
4-[(4-chloro-2-fluorophenyl)methyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
2-(4-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-1-yl)phenol
5-(2-methoxyphenoxymethyl)-N-(1,2-oxazol-3-ylmethyl)-1,2-oxazole-3-carboxamide
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[(4-methylphenyl)sulfanyl]propan-1-one
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
methyl[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl][2-(pyridin-2-yl)ethyl]amine
7-fluoro-3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)-1,2-dihydroquinolin-2-one
N3-[(3,4-dimethoxyphenyl)methyl]-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-methyl-6-(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-4-yl)pyrimidin-4-ol
(4aR,7aS)-1-acetyl-4-(naphthalen-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(diphenylmethyl)-N-[(5-methoxy-1H-indol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
7-methoxy-3-[(1-propyl-1H-pyrazol-4-yl)sulfonyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(cyclopentylmethyl)-1-(2-methoxyethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(2-methoxyphenyl)propan-1-one
1-[(2,3-dichlorophenyl)methyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
2,6-dimethyl-4-({[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]amino}methyl)phenyl acetate
4-(benzyloxy)-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]butan-1-one
(2R)-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)pyrrolidine-2-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-(1H-1,2,4-triazol-3-yl)benzamide