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N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
N'-cyclopentyl-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}butanediamide
N-[(2R)-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-1-oxopropan-2-yl]acetamide
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
7-fluoro-3-[({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amino)methyl]-1,2-dihydroquinolin-2-one
N-(3-chloro-4-fluorophenyl)-3-{1-[2-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-4-yl}propanamide
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-3-cyclopropyl-1H-pyrazole-5-carboxamide
1-[2-methoxy-6-({[3-(pyrrolidin-1-yl)propyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
(4aS,7aR)-1-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(2,4-dioxoimidazolidin-1-yl)benzamide
4-(2-hydroxybenzoyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[2-(3,4-dimethoxyphenyl)ethyl]methylamine
N-[3-(cyclohexylsulfanyl)propyl]-2-methyl-1H-1,3-benzodiazole-5-carboxamide
(1S,5R)-6-(5-chlorothiophene-2-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(3-fluorophenyl)-4-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)piperazin-2-one
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-2-oxo-N-(oxolan-2-ylmethyl)-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
1-methyl-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-chloro-4-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-dimethyl-1H-pyrazole
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-2-(piperidin-1-yl)acetamide
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-[2-({[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}amino)ethyl]acetamide
2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-methylpyridine-3-carboxylic acid
[(3-{[1-(5-chloro-3-methyl-1H-indole-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(quinolin-5-ylmethyl)amine
1-cyclopentyl-N5-[3-(dimethylamino)-2,2-dimethylpropyl]-N3,N3-diethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(2-fluorophenyl)-1-[1-(quinoxalin-6-ylmethyl)piperidin-4-yl]ethyl]-N-methylthiophene-2-carboxamide
2-{[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]methyl}pyridine-3-carboxylic acid
N-methyl-3-{methyl[(4-methyl-1H-imidazol-5-yl)methyl]amino}butanamide
(2R)-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-acetamidopropanamide
4-[2-(methylamino)-1,3-thiazole-4-carbonyl]-1-(4-methylphenyl)piperazin-2-one
1-(3-cyanopyridin-2-yl)-N-[4-(3-fluorophenyl)phenyl]piperidine-3-carboxamide
1-(2,5-dimethylphenyl)-3-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-[(3aR,6aR)-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
1-[1-({1-[2-(methylsulfanyl)benzoyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
N-[3-(3-cyano-2-methoxypyridin-4-yl)phenyl]acetamide
6-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane-11-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl]-1H-indole
3,7-dimethyl-11-[(1-phenyl-1H-pyrazol-5-yl)methyl]-3,7,11-triazaspiro[5.6]dodecane
N-(2-methoxyethyl)-4-methyl-3-{[methyl(prop-2-yn-1-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
3-(3-methoxyphenyl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
5-chloro-N-{2-[ethyl(methyl)amino]ethyl}-N-methyl-3-phenyl-1H-indole-2-carboxamide
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-(1-methyl-1H-1,2,3-benzotriazol-5-yl)urea
5-{2-[4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,3,4-thiadiazol-2-amine
ethyl 4-[4-(1H-pyrazol-4-yl)butanoyl]piperazine-1-carboxylate
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-8-(quinolin-6-yl)-1,8-diazaspiro[4.5]decane
4-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-4H-1,2,4-triazole
(5S)-5-[({[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(pyridin-2-ylmethyl)amino)methyl]pyrrolidin-2-one
(4aR,8aS)-6-(1-benzothiophen-2-ylmethyl)-1-(2-methoxyethyl)-decahydro-1,6-naphthyridin-2-one
5-[(oxolan-2-ylmethoxy)methyl]-3-(thiophen-2-yl)-1,2,4-oxadiazole