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ethyl 3-({1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(thiophen-2-yl)-1H-pyrazol-4-yl}formamido)propanoate
(1s,4s)-4-{4-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
1-[2-(3-methoxyphenyl)piperidin-1-yl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
2-(5-acetylthiophen-3-yl)-1-[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
9-methoxy-N-methyl-7-oxo-3-(quinolin-4-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-[1-methyl-5-(1,3-thiazol-4-yl)-1H-1,2,4-triazol-3-yl]pyridine
4-{[(1,2-dimethyl-1H-imidazol-5-yl)methyl]amino}-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
methyl 3-chloro-4-({4-[2-(methylsulfanyl)ethyl]piperazine-1-carbonyl}amino)benzoate
3-{5-[(6-methylpyridin-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-[(3-ethoxy-4-methoxyphenyl)methyl]-N,2-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-methyl-N-[2-(pyridin-2-yl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
(1S,5R)-6-methyl-3-{4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butanoyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
6-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1H-indole
N-{5-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazol-7-yl}acetamide
4-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-5,6,7,8-tetrahydroquinazolin-2-amine
methyl({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl){[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}amine
2-[4-(dimethylamino)phenyl]-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
(2S,4R)-N-cycloheptyl-1-{[3-(2-methylphenyl)phenyl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
(3S,4S)-1-(5-fluoropyrimidin-2-yl)-4-(naphthalen-2-yl)piperidin-3-ol
4-(furan-3-ylmethyl)-3-{2-oxo-2-[4-(thiophen-2-ylmethyl)piperazin-1-yl]ethyl}piperazin-2-one
3-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
1-ethyl-4-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1H-indole
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)pyridine-4-carboxamide
3-(4-ethyl-1H-pyrazol-5-yl)-1-[(4-fluorophenyl)methyl]piperidine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(4-methyl-1,3-thiazol-5-yl)methyl]pyrrolidin-3-yl]-5-methyl-1,2-oxazole-3-carboxamide
N-[1-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)piperidin-4-yl]methanesulfonamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-5-methyl-1H-pyrazole-3-carboxamide
ethyl 3-{[1-(2-cyclohexylethyl)-1H-1,2,3-triazol-4-yl]formamido}hexanoate
1-(1-benzoxepine-4-carbonyl)-4-(2-methoxyphenyl)-2-methylpiperazine
1-[(2-chlorophenyl)methyl]-4-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}pyrrolidin-2-one
1-[2-fluoro-3-(trifluoromethyl)phenyl]-3-[2-(pyrrolidin-1-yl)ethyl]urea
4,5-dimethyl 1-[(3S,5S)-1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-5-[(furan-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
N-ethyl-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-(2-methoxyethyl)-1-[1-(quinolin-4-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(3-propyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methanesulfonamide
2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-1,3-benzoxazole
methyl({[(1R,5S,6R)-3-(naphthalene-2-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl})(1,2-oxazol-3-ylmethyl)amine
5-methyl-N-[2-(3-methylthiophen-2-yl)ethyl]-1,3-oxazole-4-carboxamide
4-(4-chlorophenoxy)-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
7-methyl-2-(quinolin-5-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(2-methoxyphenyl)-2-[5-methyl-4-(3-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)oxane-4-carboxamide
N-(1-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-yl)methanesulfonamide
1-{3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-3-phenylprop-2-yn-1-one
5-chloro-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]thiophene-2-carboxamide
(2S)-1-[5-(6-chloro-2-fluoro-3-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]propan-2-ol
N-[(2R,3R)-2-hydroxy-1'-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
1-(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1,4-diazepan-5-one
1-[1-(8-chloroquinolin-2-yl)piperidin-4-yl]-3-methylbutan-1-ol
6-{[4-(2-propylpyrrolidine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline